Compile Data Set for Download or QSAR
Report error Found 188 Enz. Inhib. hit(s) with all data for entry = 50003659
TargetHistamine H1 receptor(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50297307(R-dimethindene | CHEMBL564226)
Affinity DataKi:  0.437nMAssay Description:Compound was evaluated for binding affinity towards cloned human histamine H1 receptors stably expressed in CHO-K1 cells using [3H]mepyramineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM81452(NSC_91533 | CAS_91533 | Dimethindene)
Affinity DataKi:  0.692nMAssay Description:Compound was evaluated for binding affinity towards cloned human histamine H1 receptors stably expressed in CHO-K1 cells using [3H]mepyramineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474506(CHEMBL167223)
Affinity DataKi:  0.813nMAssay Description:Compound was evaluated for binding affinity towards cloned human histamine H1 receptors stably expressed in CHO-K1 cells using [3H]mepyramineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474496(CHEMBL172233)
Affinity DataKi:  7.20nMAssay Description:Compound was evaluated for binding affinity towards cloned human histamine H1 receptors stably expressed in CHO-K1 cells using [3H]mepyramineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474516(CHEMBL434684)
Affinity DataKi:  12nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474489(CHEMBL423831)
Affinity DataKi:  15nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474492(CHEMBL352375)
Affinity DataKi:  25nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474492(CHEMBL352375)
Affinity DataKi:  25.1nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474489(CHEMBL423831)
Affinity DataKi:  26nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M3 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474516(CHEMBL434684)
Affinity DataKi:  29nMAssay Description:Compound was evaluated for binding affinity towards cloned human histamine H1 receptors stably expressed in CHO-K1 cells using [3H]mepyramineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474485(CHEMBL1493369)
Affinity DataKi:  30nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474496(CHEMBL172233)
Affinity DataKi:  32nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474516(CHEMBL434684)
Affinity DataKi:  32nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M3 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474506(CHEMBL167223)
Affinity DataKi:  33nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474516(CHEMBL434684)
Affinity DataKi:  35nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M1 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474497(CHEMBL171102)
Affinity DataKi:  44nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M1 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474498(CHEMBL168704)
Affinity DataKi:  45nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474490(CHEMBL171216)
Affinity DataKi:  51nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474489(CHEMBL423831)
Affinity DataKi:  52nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M1 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474497(CHEMBL171102)
Affinity DataKi:  66nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M5 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474497(CHEMBL171102)
Affinity DataKi:  68nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M3 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474485(CHEMBL1493369)
Affinity DataKi:  69nMAssay Description:Compound was evaluated for binding affinity towards cloned human histamine H1 receptors stably expressed in CHO-K1 cells using [3H]mepyramineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474489(CHEMBL423831)
Affinity DataKi:  81nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M4 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474516(CHEMBL434684)
Affinity DataKi:  87nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M5 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474506(CHEMBL167223)
Affinity DataKi:  95nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M3 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474516(CHEMBL434684)
Affinity DataKi:  98nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M4 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474486(CHEMBL354678)
Affinity DataKi:  98nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474504(CHEMBL354523)
Affinity DataKi:  107nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474488(CHEMBL353290)
Affinity DataKi:  112nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474497(CHEMBL171102)
Affinity DataKi:  129nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M4 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474485(CHEMBL1493369)
Affinity DataKi:  138nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M3 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474514(CHEMBL355769)
Affinity DataKi:  145nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474506(CHEMBL167223)
Affinity DataKi:  151nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M1 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474505(CHEMBL170221)
Affinity DataKi:  158nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M1 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474485(CHEMBL1493369)
Affinity DataKi:  191nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M1 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474492(CHEMBL352375)
Affinity DataKi:  218nMAssay Description:Compound was evaluated for binding affinity towards cloned human histamine H1 receptors stably expressed in CHO-K1 cells using [3H]mepyramineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H1 receptor(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474492(CHEMBL352375)
Affinity DataKi:  219nMAssay Description:Compound was evaluated for binding affinity towards cloned human histamine H1 receptors stably expressed in CHO-K1 cells using [3H]mepyramineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474504(CHEMBL354523)
Affinity DataKi:  224nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M1 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474497(CHEMBL171102)
Affinity DataKi:  229nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474490(CHEMBL171216)
Affinity DataKi:  229nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M1 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474493(CHEMBL169494)
Affinity DataKi:  234nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474486(CHEMBL354678)
Affinity DataKi:  240nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M1 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474499(CHEMBL170088)
Affinity DataKi:  245nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M1 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474505(CHEMBL170221)
Affinity DataKi:  257nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474488(CHEMBL353290)
Affinity DataKi:  263nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M3 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474517(CHEMBL169401)
Affinity DataKi:  263nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M2 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474504(CHEMBL354523)
Affinity DataKi:  282nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M3 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474505(CHEMBL170221)
Affinity DataKi:  288nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M3 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474485(CHEMBL1493369)
Affinity DataKi:  295nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M4 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Johannes Gutenberg-University of Mainz

Curated by ChEMBL
LigandPNGBDBM50474499(CHEMBL170088)
Affinity DataKi:  302nMAssay Description:Binding affinity towards cloned human muscarinic acetylcholine receptor M5 stably expressed in CHO-K1 cells using [3H]N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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