Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50004799
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50486005(CHEMBL2203394)
Affinity DataKd:  6.40nMAssay Description:Displacement of [3H]DMAB from amyloid beta plaque in cortex homogenate isolated from Alzheimer disease patient after 90 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485997(CHEMBL2203379)
Affinity DataKd:  4.5nMAssay Description:Displacement of [3H]DMAB from amyloid beta plaque in cortex homogenate isolated from Alzheimer disease patient after 90 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485994(CHEMBL2203385)
Affinity DataKd:  9.60nMAssay Description:Displacement of [3H]DMAB from amyloid beta plaque in cortex homogenate isolated from Alzheimer disease patient after 90 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485997(CHEMBL2203379)
Affinity DataIC50: 4nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50486007(CHEMBL2203383)
Affinity DataIC50: 8nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485994(CHEMBL2203385)
Affinity DataIC50: 11nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485999(CHEMBL2203382)
Affinity DataIC50: 14nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50486004(CHEMBL2203378)
Affinity DataIC50: 23nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50486006(CHEMBL2203384)
Affinity DataIC50: 26nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485993(CHEMBL2203387)
Affinity DataIC50: 30nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50486001(CHEMBL2203288)
Affinity DataIC50: 33nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50486000(CHEMBL2203388)
Affinity DataIC50: 36nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485995(CHEMBL2203381)
Affinity DataIC50: 42nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485992(CHEMBL2203389)
Affinity DataIC50: 45nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50486003(CHEMBL2203386)
Affinity DataIC50: 47nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485998(CHEMBL2203390)
Affinity DataIC50: 49nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485996(CHEMBL2203380)
Affinity DataIC50: 102nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50486002(CHEMBL2203392)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485991(CHEMBL2203391)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity to human amyloid beta plaqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed