Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50005904
TargetMelatonin receptor type 1B(Human)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50495327(CHEMBL3109563)
Affinity DataKi:  10nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1B(Human)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50495330(CHEMBL3109560)
Affinity DataKi:  26nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50495327(CHEMBL3109563)
Affinity DataKi:  32nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50495328(CHEMBL3109561)
Affinity DataKi:  49nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50495330(CHEMBL3109560)
Affinity DataKi:  71nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1B(Human)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50495329(CHEMBL3109562)
Affinity DataKi:  96nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50495329(CHEMBL3109562)
Affinity DataKi:  256nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1B(Human)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50495328(CHEMBL3109561)
Affinity DataKi:  315nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed