Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50007431
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063243(N-(2,6-Diisopropyl-phenyl)-2-pyridin-2-yl-malonami...)
Affinity DataIC50: 8nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLiver carboxylesterase 1(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063239(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 10nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase by microsomal LAI assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063239(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 10nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063226(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 11nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063236(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 12nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063231(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 12nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063220(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 13nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063235(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 13nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063232(2-Phenyl-N-(2,4,6-trimethoxy-phenyl)-malonamic aci...)
Affinity DataIC50: 13nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063229(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 13nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063221(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 16nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063227(2-Phenyl-N-(2,4,6-trimethoxy-phenyl)-malonamic aci...)
Affinity DataIC50: 20nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLiver carboxylesterase 1(Rabbit)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063239(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 20nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase by microsomal MAI2 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063230(N-(2,6-Diisopropyl-phenyl)-2,2-dimethyl-malonamic ...)
Affinity DataIC50: 21nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063224(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 22nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063237(2-Phenyl-N-(2,4,6-trimethoxy-phenyl)-malonamic aci...)
Affinity DataIC50: 30nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063240(N-(2,6-Diisopropyl-phenyl)-2-fluoro-malonamic acid...)
Affinity DataIC50: 32nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063233(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 37nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063234(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 40nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063222(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 50nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063225(2-Phenyl-N-(2,4,6-triisopropyl-phenyl)-malonamic a...)
Affinity DataIC50: 56nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063245(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 72nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063238(2-Pyridin-2-yl-N-(2,4,6-triisopropyl-phenyl)-malon...)
Affinity DataIC50: 180nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063223(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 200nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063242(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063228(N-(2,6-Diisopropyl-phenyl)-2-fluoro-malonamic acid...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063244(N-(2,6-Diisopropyl-phenyl)-2,2-dimethyl-malonamic ...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063241(N-(2,6-Diisopropyl-phenyl)-2-phenyl-malonamic acid...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed