Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50008024
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070169([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070180(3-(3-Hexyl-ureido)-N-(4-{2-[(S)-2-hydroxy-3-(4-hyd...)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070157(N-[4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-pr...)
Affinity DataEC50:  6.80nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070159(N-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070158(N-[4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-pr...)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070171(N-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataEC50:  1nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070160(N-[4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-pr...)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070175([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070167(4-(3-Heptyl-ureido)-N-(4-{2-[(S)-2-hydroxy-3-(4-hy...)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070176(4-(3-Hexyl-1,3-dimethyl-ureido)-N-(4-{2-[(S)-2-hyd...)
Affinity DataEC50:  10nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070170(4-(3-Hexyl-1-methyl-ureido)-N-(4-{2-[(S)-2-hydroxy...)
Affinity DataEC50:  6.60nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070172(4-(3-Cyclohexyl-ureido)-N-(4-{2-[(S)-2-hydroxy-3-(...)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070168([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070174(N-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070173([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataEC50:  11nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070164([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataEC50:  1nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070156((S)-4-(3-hexylureido)-N-(4-(2-(1-hydroxy-2-(4-hydr...)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070161(N-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataEC50:  5.20nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070179(4-(3-Hexyl-3-methyl-ureido)-N-(4-{2-[(S)-2-hydroxy...)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070163(N-[4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-pr...)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070166(Heptanoic acid [4-(4-{2-[(S)-2-hydroxy-3-(4-hydrox...)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070162(N-[4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-pr...)
Affinity DataEC50:  5nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070165(N-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070177(N-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070132(N-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070178({2-[4-(4-Amino-benzenesulfonylamino)-phenyl]-ethyl...)
Affinity DataEC50:  17nMAssay Description:Agonist activity towards human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070163(N-[4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-pr...)
Affinity DataIC50: 110nMAssay Description:In vitro affinity at Beta-2 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070173([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataIC50: 110nMAssay Description:In vitro affinity at Beta-2 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070176(4-(3-Hexyl-1,3-dimethyl-ureido)-N-(4-{2-[(S)-2-hyd...)
Affinity DataIC50: 120nMAssay Description:In vitro affinity at Beta-2 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070164([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataIC50: 130nMAssay Description:In vitro affinity at Beta-2 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070171(N-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataIC50: 150nMAssay Description:In vitro affinity at Beta-1 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070165(N-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataIC50: 150nMAssay Description:In vitro affinity at Beta-1 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070171(N-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataIC50: 170nMAssay Description:In vitro affinity at Beta-2 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070156((S)-4-(3-hexylureido)-N-(4-(2-(1-hydroxy-2-(4-hydr...)
Affinity DataIC50: 190nMAssay Description:In vitro affinity at Beta-2 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070164([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataIC50: 190nMAssay Description:In vitro affinity at Beta-1 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070173([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataIC50: 190nMAssay Description:In vitro affinity at Beta-1 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070167(4-(3-Heptyl-ureido)-N-(4-{2-[(S)-2-hydroxy-3-(4-hy...)
Affinity DataIC50: 200nMAssay Description:In vitro affinity at Beta-1 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070167(4-(3-Heptyl-ureido)-N-(4-{2-[(S)-2-hydroxy-3-(4-hy...)
Affinity DataIC50: 200nMAssay Description:In vitro affinity at Beta-2 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070156((S)-4-(3-hexylureido)-N-(4-(2-(1-hydroxy-2-(4-hydr...)
Affinity DataIC50: 200nMAssay Description:In vitro affinity at Beta-1 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070175([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataIC50: 210nMAssay Description:In vitro affinity at Beta-2 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070169([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataIC50: 220nMAssay Description:In vitro affinity at Beta-1 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070160(N-[4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-pr...)
Affinity DataIC50: 220nMAssay Description:In vitro affinity at Beta-2 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070163(N-[4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-pr...)
Affinity DataIC50: 220nMAssay Description:In vitro affinity at Beta-1 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070166(Heptanoic acid [4-(4-{2-[(S)-2-hydroxy-3-(4-hydrox...)
Affinity DataIC50: 230nMAssay Description:In vitro affinity at Beta-2 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070157(N-[4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-pr...)
Affinity DataIC50: 230nMAssay Description:In vitro affinity at Beta-2 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070175([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataIC50: 240nMAssay Description:In vitro affinity at Beta-1 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070168([4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-prop...)
Affinity DataIC50: 250nMAssay Description:In vitro affinity at Beta-1 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070172(4-(3-Cyclohexyl-ureido)-N-(4-{2-[(S)-2-hydroxy-3-(...)
Affinity DataIC50: 260nMAssay Description:In vitro affinity at Beta-1 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070170(4-(3-Hexyl-1-methyl-ureido)-N-(4-{2-[(S)-2-hydroxy...)
Affinity DataIC50: 290nMAssay Description:In vitro affinity at Beta-2 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070161(N-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propy...)
Affinity DataIC50: 300nMAssay Description:In vitro affinity at Beta-1 adrenergic receptor in the presence of [125I]iodocyanopindolol.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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