Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50010993
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50049319(N-[(R)-1-{[Acetyl-(2-methoxy-benzyl)-amino]-methyl...)
Affinity DataIC50: 0.230nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101033(N-[(R)-1-{[Acetyl-(2-methoxy-benzyl)-amino]-methyl...)
Affinity DataIC50: 0.430nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101037(N-[(R)-1-{[Acetyl-(2-methoxy-benzyl)-amino]-methyl...)
Affinity DataIC50: 0.480nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101030(N-[(R)-1-{[Acetyl-(2-chloro-benzyl)-amino]-methyl}...)
Affinity DataIC50: 0.650nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101029(1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)car...)
Affinity DataIC50: 0.820nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101031(1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)car...)
Affinity DataIC50: 0.980nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101042(1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)car...)
Affinity DataIC50: 3.20nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101034(1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)car...)
Affinity DataIC50: 3.30nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101032(1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)car...)
Affinity DataIC50: 3.5nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101035(1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)car...)
Affinity DataIC50: 6nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101040(1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)car...)
Affinity DataIC50: 8.30nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101038(1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)car...)
Affinity DataIC50: 9.70nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101041(1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)car...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101036(1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)car...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101039(1N-{2-(1H-3-indolyl)-1-[2-methoxybenzyl(methyl)car...)
Affinity DataIC50: 24nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50101028(N-[(R)-1-{[Acetyl-(2-methoxy-benzyl)-amino]-methyl...)
Affinity DataIC50: 34nMAssay Description:In vitro inhibition of binding of [125I]Bolton-Hunter SP to Tachykinin receptor 1 in human IM-9 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed