Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50011327
TargetProteinase-activated receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50105305(N-(4-{3-((R)-sec-Butyl)-3-[(S)-2-(3,4-dichloro-phe...)
Affinity DataIC50: 120nMAssay Description:Binding affinity against platelet thrombin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50105328(N-(4-{3-[(S)-2-(3,4-Dichloro-phenyl)-2-hydroxy-eth...)
Affinity DataIC50: 700nMAssay Description:Binding affinity against platelet thrombin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50105336((2S,5S)-2-[(S)-(3,4-Dichloro-phenyl)-hydroxy-methy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity against platelet thrombin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50105338((S)-2-[(S)-(3,4-Dichloro-phenyl)-hydroxy-methyl]-p...)
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity against platelet thrombin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50105311(N-(4-{3-[(S)-2-(3,4-Dichloro-phenyl)-2-hydroxy-eth...)
Affinity DataIC50: 1.20E+3nMAssay Description:Binding affinity against platelet thrombin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50105321(N-(4-{3-Cyclopropyl-3-[(S)-2-(3,4-dichloro-phenyl)...)
Affinity DataIC50: 2.10E+3nMAssay Description:Binding affinity against platelet thrombin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50105352(N-(4-{3-[(S)-2-(3,4-Dichloro-phenyl)-2-hydroxy-eth...)
Affinity DataIC50: 6.60E+3nMAssay Description:Binding affinity against platelet thrombin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed