Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50011405
LigandPNGBDBM50106179(Enantiomer-4-(3-Butyl-[1,2,4]oxadiazol-5-yl)-N-(2,...)
Affinity DataIC50: 2nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50106169(Enantiomer-4-(3-Butyl-[1,2,4]oxadiazol-5-yl)-N-(2,...)
Affinity DataIC50: 9nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50106167(Enantiomer-4-(3-Cyclopropylmethyl-[1,2,4]oxadiazol...)
Affinity DataIC50: 18nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50106167(Enantiomer-4-(3-Cyclopropylmethyl-[1,2,4]oxadiazol...)
Affinity DataIC50: 18nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106178(4-(3-Butyl-[1,2,4]oxadiazol-5-yl)-N-(3,3-dimethyl-...)
Affinity DataIC50: 23nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50106168(Enantiomer-N-(2,2-Dimethyl-cyclopentylmethyl)-4-(3...)
Affinity DataIC50: 27nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106168(Enantiomer-N-(2,2-Dimethyl-cyclopentylmethyl)-4-(3...)
Affinity DataIC50: 27nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50061218((E)-3-(2,4-Dichloro-phenyl)-N-((R)-1-methyl-2-oxo-...)
Affinity DataIC50: 31nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106176(Enantiomer-N-(2,2-Dimethyl-cyclopentylmethyl)-4-[5...)
Affinity DataIC50: 40nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106176(Enantiomer-N-(2,2-Dimethyl-cyclopentylmethyl)-4-[5...)
Affinity DataIC50: 40nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106182(N-(3,3-Dimethyl-butyl)-4-(3-phenyl-[1,2,4]oxadiazo...)
Affinity DataIC50: 130nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106166(N-(3,3-Dimethyl-butyl)-4-hexyloxy-benzamide | CHEM...)
Affinity DataIC50: 250nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106177(N-(3,3-Dimethyl-butyl)-4-indol-1-yl-benzamide | CH...)
Affinity DataIC50: 260nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106184(N-(3,3-Dimethyl-cyclopentyl)-4-hexyloxy-benzamide ...)
Affinity DataIC50: 360nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106180(N-(3,3-Dimethyl-cyclohexylmethyl)-4-hexyloxy-benza...)
Affinity DataIC50: 370nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106181(Biphenyl-4-carboxylic acid (3,3-dimethyl-butyl)-am...)
Affinity DataIC50: 540nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106164(Enantiomer-N-(2,2-Dimethyl-cyclopentylmethyl)-4-(3...)
Affinity DataIC50: 580nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106164(Enantiomer-N-(2,2-Dimethyl-cyclopentylmethyl)-4-(3...)
Affinity DataIC50: 580nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106175(Enantiomer-N-(2,2-Dimethyl-cyclopentylmethyl)-4-he...)
Affinity DataIC50: 710nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106175(Enantiomer-N-(2,2-Dimethyl-cyclopentylmethyl)-4-he...)
Affinity DataIC50: 710nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106174(N-(2,2-Dimethyl-cyclohexylmethyl)-4-hexyloxy-benza...)
Affinity DataIC50: 1.40E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106165((3-tert-Butyl-pyrrolidin-1-yl)-(4-hexyloxy-phenyl)...)
Affinity DataIC50: 3.00E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106174(N-(2,2-Dimethyl-cyclohexylmethyl)-4-hexyloxy-benza...)
Affinity DataIC50: 3.00E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106170(N-(2-Diethylamino-ethyl)-4-hexyloxy-benzamide | CH...)
Affinity DataIC50: 3.50E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106183(1-(4-Hexyloxy-phenyl)-3-piperidin-1-yl-propan-1-on...)
Affinity DataIC50: 4.00E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106173(N,N-Diethyl-2-[4-(1,1,3,3-tetramethyl-butyl)-pheno...)
Affinity DataIC50: 5.00E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106171(Diethyl-{2-[4-(1,1,3,3-tetramethyl-butyl)-phenoxy]...)
Affinity DataIC50: 5.00E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50106172(N-(2,2-Dimethyl-cyclopentyl)-4-hexyloxy-benzamide ...)
Affinity DataIC50: 3.00E+4nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricular myocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed