Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50013288
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128682(N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-(4-diethylamin...)
Affinity DataIC50: 700nMAssay Description:Inhibition of degradation of tyrosine kinase pp60src by Calpain 1 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50073850([(S)-1-(1-Benzyl-2-oxo-ethylcarbamoyl)-2-methyl-pr...)
Affinity DataIC50: 700nMAssay Description:Inhibition of degradation of tyrosine kinase pp60src by Calpain 1 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128679(N-(1-Carbamoyl-pentyl)-2-[2-(4-dimethylaminomethyl...)
Affinity DataIC50: 800nMAssay Description:Inhibition of degradation of tyrosine kinase pp60src by Calpain 1 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128681(N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-(4-dimethylami...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of degradation of tyrosine kinase pp60src by Calpain 1 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128678(N-(1-Carbamoyl-2-phenyl-ethyl)-2-(2-naphthalen-1-y...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of degradation of tyrosine kinase pp60src by Calpain 1 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128678(N-(1-Carbamoyl-2-phenyl-ethyl)-2-(2-naphthalen-1-y...)
Affinity DataKi:  8.40nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128679(N-(1-Carbamoyl-pentyl)-2-[2-(4-dimethylaminomethyl...)
Affinity DataKi:  13.3nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128680(N-(1-Benzyl-2-oxo-ethyl)-2-(2-naphthalen-1-yl-viny...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50073850([(S)-1-(1-Benzyl-2-oxo-ethylcarbamoyl)-2-methyl-pr...)
Affinity DataKi:  15.5nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50073850([(S)-1-(1-Benzyl-2-oxo-ethylcarbamoyl)-2-methyl-pr...)
Affinity DataKi:  18nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128681(N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-(4-dimethylami...)
Affinity DataKi:  18.3nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128682(N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-(4-diethylamin...)
Affinity DataKi:  27nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128679(N-(1-Carbamoyl-pentyl)-2-[2-(4-dimethylaminomethyl...)
Affinity DataKi:  27nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128682(N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-(4-diethylamin...)
Affinity DataKi:  62nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128681(N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-(4-dimethylami...)
Affinity DataKi:  83nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCathepsin B(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50128678(N-(1-Carbamoyl-2-phenyl-ethyl)-2-(2-naphthalen-1-y...)
Affinity DataKi:  99nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50112839(N-(1-Benzyl-2-oxo-ethyl)-2-styryl-benzamide | CHEM...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Abbott

Curated by ChEMBL
LigandPNGBDBM50112838(N-(1-Benzyl-2-oxo-ethyl)-benzamide | CHEMBL281874)
Affinity DataKi:  1.08E+3nMAssay Description:Inhibitory activity against human Calpain 1 isolated from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed