Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50043541
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442711(CHEMBL2442509)
Affinity DataIC50: 10nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442711(CHEMBL2442509)
Affinity DataIC50: 59nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442710(CHEMBL1303766)
Affinity DataIC50: 250nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442718(CHEMBL2442512)
Affinity DataIC50: 730nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442710(CHEMBL1303766)
Affinity DataIC50: 860nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442717(CHEMBL2442515)
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442716(CHEMBL2442510)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442715(CHEMBL2442513)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442714(CHEMBL1830821)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442713(CHEMBL2442514)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442712(CHEMBL2442508)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442701(CHEMBL2074836)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442702(CHEMBL2442511 | US9296728, 26)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442709(CHEMBL2442516)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442708(CHEMBL2442517)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442707(CHEMBL2442503)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442706(CHEMBL2442504)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442705(CHEMBL2442505)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442704(CHEMBL2442506)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442703(CHEMBL2442507)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMonocarboxylate transporter 4(Human)
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442701(CHEMBL2074836)
Affinity DataIC50: 4.35E+4nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed