Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50048758
LigandPNGBDBM50226906(CHEMBL30001)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of canine cardiac fraction III cAMP phosphodiesterase (PDE 3) at 1.875 mg/kg intravenous doseMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50226909(CHEMBL31133)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibitory activity against canine cardiac fraction III cyclic AMP phosphodiesterase (PDE III) at 8.75 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226910(Bemarinone)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of canine cardiac fraction III cAMP phosphodiesterase (PDE 3) at 0.875 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226905(CHEMBL1743762)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibitory activity against canine cardiac fraction III cyclic AMP phosphodiesterase (PDE III) at 8.75 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226908(CHEMBL30387)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of canine cardiac fraction III cAMP phosphodiesterase (PDE 3) at 1.875 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226907(CHEMBL30636)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibitory activity against canine cardiac fraction III cyclic AMP phosphodiesterase (PDE III) at 8.75 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226913(CHEMBL30542)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against canine cardiac fraction III cyclic AMP phosphodiesterase (PDE III) at 8.75 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226912(CHEMBL284443)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibitory activity against canine cardiac fraction III cyclic AMP phosphodiesterase (PDE III) at 8.75 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226914(CHEMBL30607)
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibitory activity against canine cardiac fraction III cyclic AMP phosphodiesterase (PDE III) at 8.75 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM34651(MLS000069829 | cid_3698 | SMR000058850 | CHEMBL128...)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of canine cardiac fraction III cAMP phosphodiesterase (PDE 3) at 1.875 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226903(CHEMBL30699)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against canine cardiac fraction III cyclic AMP phosphodiesterase (PDE III) at 8.75 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226915(CHEMBL284798)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against canine cardiac fraction III cyclic AMP phosphodiesterase (PDE III) at 8.75 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226904(CHEMBL30629)
Affinity DataIC50: 1.29E+5nMAssay Description:Inhibitory activity against canine cardiac fraction III cyclic AMP phosphodiesterase (PDE III) at 8.75 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226916(CHEMBL281242)
Affinity DataIC50: 1.38E+5nMAssay Description:Inhibitory activity against canine cardiac fraction III cyclic AMP phosphodiesterase (PDE III) at 8.75 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226911(CHEMBL30541)
Affinity DataIC50: 1.90E+5nMAssay Description:Inhibitory activity against canine cardiac fraction III cyclic AMP phosphodiesterase (PDE III) at 8.75 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50226902(CHEMBL435758)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of canine cardiac fraction III cAMP phosphodiesterase (PDE 3) at 1.875 mg/kg intravenous doseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed