Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 5353
TargetNorepinephrine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM35229(Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[...)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetNorepinephrine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  0.460nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM25870(CITALOPRAM HYDROBROMIDE | [3H]Escitalopram | Escit...)
Affinity DataKi:  0.820nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM50028091((1E)-5-methoxy-1-[4-(trifluoromethyl)phenyl]pentan...)
Affinity DataKi:  2.77nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetSodium-dependent dopamine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM50021952(CHEMBL35337 | 7-Benzyl-1-ethyl-4-oxo-1,4-dihydro-[...)
Affinity DataKi:  18.7nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  52.8nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM50062915(methyl (2R)-phenyl[(2R)-piperidin-2-yl]acetate | m...)
Affinity DataKi:  125nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetNorepinephrine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM50062915(methyl (2R)-phenyl[(2R)-piperidin-2-yl]acetate | m...)
Affinity DataKi:  126nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  158nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM35229(Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[...)
Affinity DataKi:  228nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM22417(LY 94939 | Nisoxetine Inhibitor | Nisoxetine | LY1...)
Affinity DataKi:  505nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNorepinephrine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNorepinephrine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM50028091((1E)-5-methoxy-1-[4-(trifluoromethyl)phenyl]pentan...)
Affinity DataKi:  5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNorepinephrine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNorepinephrine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM25870(CITALOPRAM HYDROBROMIDE | [3H]Escitalopram | Escit...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNorepinephrine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM50021952(CHEMBL35337 | 7-Benzyl-1-ethyl-4-oxo-1,4-dihydro-[...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM50028091((1E)-5-methoxy-1-[4-(trifluoromethyl)phenyl]pentan...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM35229(Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM25870(CITALOPRAM HYDROBROMIDE | [3H]Escitalopram | Escit...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Harvard University

Curated by PDSP Ki Database
LigandPNGBDBM50062915(methyl (2R)-phenyl[(2R)-piperidin-2-yl]acetate | m...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed