Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 452
LigandChemical structure of BindingDB Monomer ID 2685BDBM2685(3-(1H-indol-3-yl)-4-{1-[2-(piperidin-2-yl)ethyl]-1...)
Affinity DataIC50: 5nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
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Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2683BDBM2683(2-[1-(3-dimethylaminopropyl)-indol-3-yl]-3-(indol-...)
Affinity DataIC50: 10nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
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Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2694BDBM2694(3-(1H-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl...)
Affinity DataIC50: 13nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
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Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2691BDBM2691(Bisindolyl deriv. 19 | 3-[1-(3-aminopropyl)-1H-ind...)
Affinity DataIC50: 26nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
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Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2681BDBM2681(3-{1-[3-(dimethylamino)propyl]-1H-indol-3-yl}-4-(1...)
Affinity DataIC50: 40nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2692BDBM2692(3-(1H-indol-3-yl)-4-{1-[(1-methylpiperidin-3-yl)me...)
Affinity DataIC50: 45nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
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Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2686BDBM2686(3-(1H-indol-3-yl)-4-{1-[3-(piperazin-1-yl)propyl]-...)
Affinity DataIC50: 52nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2693BDBM2693(3-(1H-indol-3-yl)-4-{1-[3-(morpholin-4-yl)propyl]-...)
Affinity DataIC50: 70nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2690BDBM2690(3-(1-{2-[(dimethylamino)methyl]propyl}-1H-indol-3-...)
Affinity DataIC50: 80nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2682BDBM2682(3-{1-[3-(dimethylamino)propyl]-1H-indol-3-yl}-4-[1...)
Affinity DataIC50: 100nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2583BDBM2583(bis-indolylmaleimide deriv. 8a | 3,4-bis(1H-indol-...)
Affinity DataIC50: 100nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2687BDBM2687(methyl 3-{3-[4-(1H-indol-3-yl)-2,5-dioxo-2,5-dihyd...)
Affinity DataIC50: 200nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2688BDBM2688(3-(1H-indol-3-yl)-4-[1-(2-methoxyethyl)-1H-indol-3...)
Affinity DataIC50: 200nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2680BDBM2680(3-(6-hydroxy-1H-indol-3-yl)-4-(1H-indol-3-yl)-2,5-...)
Affinity DataIC50: 200nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2684BDBM2684(indolocarbazole deriv. 4f | 3-[3-(dimethylamino)pr...)
Affinity DataIC50: 260nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2586BDBM2586(3,4-bis(1H-indol-3-yl)-2,5-dihydro-1H-pyrrol-2-one...)
Affinity DataIC50: 2.00E+3nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2689BDBM2689(3-[1-(3-dymethylaminopropyl)-indol-3-yl]-4-(indol-...)
Affinity DataIC50: 2.75E+3nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2676BDBM2676(3,4-bis(1H-indol-3-yl)pyrrolidine-2,5-dione | Bisi...)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2587BDBM2587(5-Hydroxy-3,4-Bis(3-indolyl)-3-pyrrolin-2-one | Bi...)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2679BDBM2679(3,4-bis(2-methyl-1H-indol-3-yl)-2,5-dihydro-1H-pyr...)
Affinity DataIC50: 2.00E+4nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2581BDBM2581(CHEMBL16958 | 3,13,23-triazahexacyclo[14.7.0.0^{2,...)
Affinity DataIC50: 2.50E+4nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2672BDBM2672(6,7,12,13-Tetrahydro-5,7-dioxo-5H-indolo[2,3-a]pyr...)
Affinity DataIC50: 4.00E+4nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2582BDBM2582(CHEMBL291725 | 3,4-bis(1H-indol-3-yl)-1-methyl-2,5...)
Affinity DataIC50: 5.00E+4nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 2588BDBM2588(3,4-bis(1H-indol-3-yl)-2,5-dihydrofuran-2,5-dione ...)
Affinity DataIC50: 5.00E+4nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2004
Entry Details
PubMed