Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50001521
TargetAdenosine receptor A2b(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258672BDBM50258672([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  0.794nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282641BDBM50282641(CHEMBL4160732)
Affinity DataKi:  1nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282638BDBM50282638(CHEMBL4175851)
Affinity DataKi:  1.30nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282631BDBM50282631(CHEMBL4175454)
Affinity DataKi:  1.80nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50233089BDBM50233089(8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-...)
Affinity DataKi:  6nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282640BDBM50282640(CHEMBL4168653)
Affinity DataEC50:  17nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086170BDBM50086170(CHEMBL1628266 | N-(4-Cyano-phenyl)-2-[4-(2,6-dioxo...)
Affinity DataEC50:  23nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282639BDBM50282639(CHEMBL4165135)
Affinity DataEC50:  23nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282637BDBM50282637(CHEMBL4167064)
Affinity DataEC50:  35nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282636BDBM50282636(CHEMBL4163380)
Affinity DataEC50:  35nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282642BDBM50282642(CHEMBL4173768)
Affinity DataEC50:  47nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/1/2020
Entry Details Article
PubMed