Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50040086
TargetE3 ubiquitin-protein ligase XIAP(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50388975BDBM50388975(CHEMBL2063869)
Affinity DataKi:  28nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50388974BDBM50388974(CHEMBL2063868)
Affinity DataKi:  35nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50388970BDBM50388970(CHEMBL2063863)
Affinity DataKi:  190nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50388968BDBM50388968(CHEMBL2063866)
Affinity DataKi:  410nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50388969BDBM50388969(CHEMBL2063862)
Affinity DataKi:  430nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50388973BDBM50388973(CHEMBL2063867)
Affinity DataKi:  700nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50388972BDBM50388972(CHEMBL2063865)
Affinity DataKi:  800nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50388971BDBM50388971(CHEMBL2063864)
Affinity DataKi:  7.60E+3nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed