Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 2139
LigandChemical structure of BindingDB Monomer ID 17290BDBM17290(EM1745 | E2-adenosine hybrid compound, 8 | [5-(6-a...)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/molepH: 7.5 T: 2°CAssay Description:For steady-state kinetic study of hybrid inhibitors, a Fluorolog 3 instrument was used to monitor the fluorescent signal of NADPH formed during estra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 17293BDBM17293([5-(6-amino-9H-purin-9-yl)-3,4-dihydroxyoxolan-2-y...)
Affinity DataKi:  2.50E+5nM ΔG°:  -21.4kJ/molepH: 7.5 T: 2°CAssay Description:For steady-state kinetic study of hybrid inhibitors, a Fluorolog 3 instrument was used to monitor the fluorescent signal of NADPH formed during estra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 17294BDBM17294(Compound 11 | (13S,14S,15S)-15-methyl-13-nonyltetr...)
Affinity DatapH: 7.5 T: 2°CAssay Description:For steady-state kinetic study of hybrid inhibitors, a Fluorolog 3 instrument was used to monitor the fluorescent signal of NADPH formed during estra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2007
Entry Details Article
PubMed