Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50001489
TargetVitamin D3 receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.0700nMAssay Description:Transactivation of VP16-tagged VDR (unknown origin) expressed in HEK293 cells harboring pCMX-GAL4-RXRalpha and MH100(UAS) X 4tk-LUC reporter plasmid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50281390(CHEMBL4159525)
Affinity DataEC50:  0.140nMAssay Description:Transactivation of VP16-tagged VDR (unknown origin) expressed in HEK293 cells harboring pCMX-GAL4-RXRalpha and MH100(UAS) X 4tk-LUC reporter plasmid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50281389(CHEMBL4173602)
Affinity DataEC50: >1.20nMAssay Description:Transactivation of VP16-tagged VDR (unknown origin) expressed in HEK293 cells harboring pCMX-GAL4-RXRalpha and MH100(UAS) X 4tk-LUC reporter plasmid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2020
Entry Details Article
PubMed