Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50047668
TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50182282BDBM50182282(CHEMBL3818905)
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2017
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50182281BDBM50182281(CHEMBL3818205)
Affinity DataIC50: 70nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2017
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50182283BDBM50182283(CHEMBL3819313)
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2017
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50182284BDBM50182284(CHEMBL3818888)
Affinity DataIC50: 250nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2017
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81818BDBM81818(CHEMBL1909810 | NSC_1794 | CAS_1794 | HMA)
Affinity DataIC50: 270nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2017
Entry Details Article
PubMed