Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 7602
TargetBromodomain-containing protein 3 [306-416](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.00270nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4 [333-460](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.00430nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 2 [348-455](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.00690nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.00780nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 2 [71-194,348-455](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.0100nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4 [44-168,333-460](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.0120nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 3 [24-144,306-416](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0120nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 2 [71-194](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.0140nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 2 [71-194,348-455](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0240nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 2 [348-455](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0330nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4 [333-460](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0530nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 3 [24-144](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0590nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0620nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [251-382](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.0660nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 3 [306-416](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0700nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137,251-382](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0760nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [251-382](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0860nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4 [44-168,333-460](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0870nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4 [44-168](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0990nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 3 [24-144,306-416](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.110nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 3 [24-144](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.130nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 2 [71-194](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.160nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4 [44-168](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.180nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.290nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137,251-382](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.420nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.560nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 2 [71-194,348-455](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  5.60nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4 [44-168,333-460](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  7.30nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4 [333-460](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  8.20nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetIsoform C of Bromodomain-containing protein 4 (Short)(Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  11nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 3 [24-144,306-416](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  14nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 4 [44-168](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  14nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 3 [24-144](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  14nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 2 [348-455](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  18nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 3 [306-416](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  19nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain-containing protein 2 [71-194](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  27nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [251-382](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  35nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137,251-382](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  46nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205429BDBM205429( (R)-JQ1 (3) | US9320741, (R)-JQ1 | US10407441, Co...)
Affinity DataKd:  47nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed