Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataKi: 99nMpH: 7.4Assay Description:Membranes prepared as above were resuspended to 1 ug protein/ul (measured by Bradford assay using BSA as standard), and 50 ul were added to each well...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataKi: 115nMpH: 7.4Assay Description:Membranes prepared as above were resuspended to 1 ug protein/ul (measured by Bradford assay using BSA as standard), and 50 ul were added to each well...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataKi: 124nM ΔG°: -39.0kJ/molepH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataKi: 250nMpH: 7.4Assay Description:Membranes prepared as above were resuspended to 1 ug protein/ul (measured by Bradford assay using BSA as standard), and 50 ul were added to each well...More data for this Ligand-Target Pair
Affinity DataKi: 1.11E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional
receptor assays are available on the NIMH PDSP website at
http://pdsp.med.un...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataKi: >2.00E+3nM ΔG°: >-32.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein (obtained from cells expressing the receptor) and test compo...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataKi: >2.00E+3nM ΔG°: >-32.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein (obtained from cells expressing the receptor) and test compo...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataKi: >2.00E+3nM ΔG°: >-32.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein (obtained from cells expressing the receptor) and test compo...More data for this Ligand-Target Pair
Affinity DataKi: 3.39E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional
receptor assays are available on the NIMH PDSP website at
http://pdsp.med.un...More data for this Ligand-Target Pair
Affinity DataKi: 3.76E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional
receptor assays are available on the NIMH PDSP website at
http://pdsp.med.un...More data for this Ligand-Target Pair
Affinity DataKi: 6.37E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional
receptor assays are available on the NIMH PDSP website at
http://pdsp.med.un...More data for this Ligand-Target Pair
Affinity DataKi: 6.74E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional
receptor assays are available on the NIMH PDSP website at
http://pdsp.med.un...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 12.1nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 14.6nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 25.5nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 27nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 34.6nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 37.4nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 37.9nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 39nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 46nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 50.8nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 59nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 62nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 63nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 66nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 71nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 76.6nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 78.1nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 88nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 93.6nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 94.3nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 101nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 103nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 109nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 127nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 130nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 136nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 140nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 146nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 146nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 146nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 159nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 189nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 193nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 200nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 204nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 207nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 227nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Carolina At Chapel Hill
US Patent
University Of North Carolina At Chapel Hill
US Patent
Affinity DataIC50: 290nMpH: 7.4Assay Description:For serotonin 5-HT2A binding, an aliquot of human recombinant serotonin 5-HT2A receptor (PerkinElmer Life and Analytical Sciences, USA) expressed in ...More data for this Ligand-Target Pair