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Found 7 of ph data with Target = '5-hydroxytryptamine receptor 4'
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs

LigandPNGBDBM29531(ML10302 scaffold, 9{b;w})
Affinity DataKi:  2nM ΔG°:  -49.7kJ/mole EC50:  68nMpH: 7.4 T: 2°CAssay Description:Radioligand binding studies were performed in buffer contains test compound, [3H]-GR113808, and receptor C6 glial cell membrane preparation. Nonspeci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs

LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  5nM ΔG°:  -47.4kJ/mole EC50:  51nMpH: 7.4 T: 2°CAssay Description:Radioligand binding studies were performed in buffer contains test compound, [3H]-GR113808, and receptor C6 glial cell membrane preparation. Nonspeci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs

LigandPNGBDBM29527(ML10302 scaffold, 9{a;q})
Affinity DataKi:  5nM ΔG°:  -47.4kJ/mole EC50:  18nMpH: 7.4 T: 2°CAssay Description:Radioligand binding studies were performed in buffer contains test compound, [3H]-GR113808, and receptor C6 glial cell membrane preparation. Nonspeci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs

LigandPNGBDBM29530(ML10302 scaffold, 19)
Affinity DataKi:  12nM ΔG°:  -45.2kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding studies were performed in buffer contains test compound, [3H]-GR113808, and receptor C6 glial cell membrane preparation. Nonspeci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs

LigandPNGBDBM29529(ML10302 scaffold, 14)
Affinity DataKi:  14nM ΔG°:  -44.8kJ/mole EC50:  9nMpH: 7.4 T: 2°CAssay Description:Radioligand binding studies were performed in buffer contains test compound, [3H]-GR113808, and receptor C6 glial cell membrane preparation. Nonspeci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs

LigandPNGBDBM29528(ML10302 scaffold, 9{a;y})
Affinity DataKi:  111nM ΔG°:  -39.7kJ/mole EC50:  4nMpH: 7.4 T: 2°CAssay Description:Radioligand binding studies were performed in buffer contains test compound, [3H]-GR113808, and receptor C6 glial cell membrane preparation. Nonspeci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs

LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi:  1.05E+3nM ΔG°:  -34.1kJ/mole EC50:  12nMpH: 7.4 T: 2°CAssay Description:Radioligand binding studies were performed in buffer contains test compound, [3H]-GR113808, and receptor C6 glial cell membrane preparation. Nonspeci...More data for this Ligand-Target Pair