Compile Data Set for Download or QSAR
Report error Found 182 of ph data with Target = 'Adenosine receptor A1'
TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191826BDBM191826(US9187428, 54)
Affinity DataEC50:  0.0400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191818BDBM191818(US9187428, 46)
Affinity DataEC50:  0.0400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191778BDBM191778(US9187428, 6)
Affinity DataEC50:  0.0600nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191785BDBM191785(US9187428, 13)
Affinity DataEC50:  0.0800nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191850BDBM191850(US9187428, 78)
Affinity DataEC50:  0.100nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191779BDBM191779(US9187428, 7)
Affinity DataEC50:  0.100nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191798BDBM191798(US9187428, 26)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191854BDBM191854(US9187428, 82)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191823BDBM191823(US9187428, 51)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191855BDBM191855(US9187428, 83)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191775BDBM191775(US9187428, 3)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191842BDBM191842(US9187428, 70)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191873BDBM191873(US9187428, 101)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191847BDBM191847(US9187428, 75)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191866BDBM191866(US9187428, 94)
Affinity DataEC50:  0.200nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191799BDBM191799(US9187428, 27)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191821BDBM191821(US9187428, 49)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191776BDBM191776(US9187428, 53 | US9187428, 4)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191776BDBM191776(US9187428, 53 | US9187428, 4)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191834BDBM191834(US9187428, 62)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191774BDBM191774(US9187428, 2)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191805BDBM191805(US9187428, 33)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191870BDBM191870(US9187428, 98)
Affinity DataEC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191827BDBM191827(US9187428, 55)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191832BDBM191832(US9187428, 60)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191800BDBM191800(US9187428, 28)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191856BDBM191856(US9187428, 84)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191816BDBM191816(US9187428, 44)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191868BDBM191868(US9187428, 96)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191802BDBM191802(US9187428, 30)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191840BDBM191840(US9187428, 68)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191804BDBM191804(US9187428, 32)
Affinity DataEC50:  0.400nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 21173BDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  0.5nM ΔG°:  -53.1kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191857BDBM191857(US9187428, 85)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191801BDBM191801(US9187428, 29)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191822BDBM191822(US9187428, 50)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191810BDBM191810(US9187428, 38)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191844BDBM191844(US9187428, 72)
Affinity DataEC50:  0.5nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 21173BDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  0.5nM ΔG°:  -53.1kJ/molepH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (30 ug proteins) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 2 mM MgCl2, 2 units/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 21216BDBM21216(2-[4-(ethylsulfanyl)-1H-1,3-benzodiazol-2-yl]quino...)
Affinity DataKi:  0.5nM ΔG°:  -53.1kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191859BDBM191859(US9187428, 87)
Affinity DataEC50:  0.600nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191860BDBM191860(US9187428, 88)
Affinity DataEC50:  0.700nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191809BDBM191809(US9187428, 37)
Affinity DataEC50:  0.700nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191787BDBM191787(US9187428, 15)
Affinity DataEC50:  0.800nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 50085658BDBM50085658(2-Cl-CPA | CHEMBL284969 | 2-chloro-N6-cyclopentyla...)
Affinity DataKi:  0.830nM ΔG°:  -48.2kJ/molepH: 7.4 T: 2°CAssay Description:Membranes for radioligand binding experiments are prepared from fresh or frozen cells as described in Klotz et al., Naunyn-Schmiedeberg's Arch. Pharm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2013
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191865BDBM191865(US9187428, 93)
Affinity DataEC50:  0.900nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191793BDBM191793(US9187428, 21)
Affinity DataEC50:  0.900nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191871BDBM191871(US9187428, 99)
Affinity DataEC50:  0.900nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 97464BDBM97464(US8609833, 17 | US8470800, A | US8609833, 86)
Affinity DataKi:  0.970nM ΔG°:  -47.8kJ/molepH: 7.4 T: 2°CAssay Description:Membranes for radioligand binding experiments are prepared from fresh or frozen cells as described in Klotz et al., Naunyn-Schmiedeberg's Arch. Pharm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2013
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Bayer Intellectual Property

US Patent
LigandChemical structure of BindingDB Monomer ID 191838BDBM191838(US9187428, 66)
Affinity DataEC50:  1.30nMpH: 7.4 T: 2°CAssay Description:The stock cultures are grown, at 37° C. and under 5% CO2, in DMEM/F12 medium containing 10% FCS (fetal calf serum) and in each case split 1:10 af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2016
Entry Details
US Patent

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