Compile Data Set for Download or QSAR
Report error Found 35 of ph data with Target = 'Alpha-mannosidase 2'
TargetAlpha-mannosidase 2(Fruit fly)
University of Toronto

LigandPNGBDBM84871(Swainsonine derivative, 6)
Affinity DataIC50: 44nMpH: 5.75 T: 2°CAssay Description:Inhibition of dGMII was measured at pH 5.75. Determination of the IC50 values (concentrations of inhibitor at which 50% of activity remains) was car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Fruit fly)
University of Toronto

LigandPNGBDBM84872(Swainsonine derivative, 7)
Affinity DataIC50: 250nMpH: 5.75 T: 2°CAssay Description:Inhibition of dGMII was measured at pH 5.75. Determination of the IC50 values (concentrations of inhibitor at which 50% of activity remains) was car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Fruit fly)
University of Toronto

LigandPNGBDBM84870(Swainsonine derivative, 5)
Affinity DataIC50: 250nMpH: 5.75 T: 2°CAssay Description:Inhibition of dGMII was measured at pH 5.75. Determination of the IC50 values (concentrations of inhibitor at which 50% of activity remains) was car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Fruit fly)
University of Toronto

LigandPNGBDBM84869(Swainsonine derivative, 4)
Affinity DataKi:  2.70nM ΔG°:  -48.9kJ/mole IC50: 29nMpH: 5.75 T: 2°CAssay Description:Inhibition of dGMII was measured at pH 5.75. Determination of the IC50 values (concentrations of inhibitor at which 50% of activity remains) was car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Fruit fly)
University of Toronto

LigandPNGBDBM84868(Swainsonine derivative, 3)
Affinity DataKi:  2.70nM ΔG°:  -48.9kJ/mole IC50: 29nMpH: 5.75 T: 2°CAssay Description:Inhibition of dGMII was measured at pH 5.75. Determination of the IC50 values (concentrations of inhibitor at which 50% of activity remains) was car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Fruit fly)
University of Toronto

LigandPNGBDBM84867(Swainsonine derivative, 2)
Affinity DataKi:  2.80nM ΔG°:  -48.8kJ/mole IC50: 30nMpH: 5.75 T: 2°CAssay Description:Inhibition of dGMII was measured at pH 5.75. Determination of the IC50 values (concentrations of inhibitor at which 50% of activity remains) was car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Fruit fly)
University of Toronto

LigandPNGBDBM50168995((-)-swainsonine | CHEMBL371197 | (1S,2R,8R,8aR)-Oc...)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/mole IC50: 37nMpH: 5.75 T: 2°CAssay Description:Inhibition of dGMII was measured at pH 5.75. Determination of the IC50 values (concentrations of inhibitor at which 50% of activity remains) was car...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84465(Benzylation of mannostatin A, 1e)
Affinity DataKi:  50nM ΔG°:  -43.3kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM50078117(Mannostatin A, 1 | (1R,2R,3R,4S,5R)-4-Amino-5-meth...)
Affinity DataKi:  90nM ΔG°:  -41.8kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84464(Benzylation of mannostatin A, 1d)
Affinity DataKi:  100nM ΔG°:  -41.6kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84466(Benzylation of mannostatin A, 1f)
Affinity DataKi:  100nM ΔG°:  -41.6kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84462(Benzylation of mannostatin A, 1b)
Affinity DataKi:  110nM ΔG°:  -41.3kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84467(Benzylation of mannostatin A, 1g)
Affinity DataKi:  140nM ΔG°:  -40.7kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84474(Aminocyclopentitetrol, 2g)
Affinity DataKi:  160nM ΔG°:  -40.3kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84463(Benzylation of mannostatin A, 1c)
Affinity DataKi:  170nM ΔG°:  -40.2kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM50078117(Mannostatin A, 1 | (1R,2R,3R,4S,5R)-4-Amino-5-meth...)
Affinity DataKi:  210nM ΔG°:  -39.6kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84472(Aminocyclopentitetrol, 2e)
Affinity DataKi:  330nM ΔG°:  -38.5kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84470(Aminocyclopentitetrol, 2c)
Affinity DataKi:  330nM ΔG°:  -38.5kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84469(Aminocyclopentitetrol, 2b)
Affinity DataKi:  450nM ΔG°:  -37.7kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84473(Aminocyclopentitetrol, 2f)
Affinity DataKi:  480nM ΔG°:  -37.5kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84465(Benzylation of mannostatin A, 1e)
Affinity DataKi:  510nM ΔG°:  -37.4kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84466(Benzylation of mannostatin A, 1f)
Affinity DataKi:  520nM ΔG°:  -37.3kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84463(Benzylation of mannostatin A, 1c)
Affinity DataKi:  530nM ΔG°:  -37.3kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84471(Aminocyclopentitetrol, 2d)
Affinity DataKi:  670nM ΔG°:  -36.7kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84462(Benzylation of mannostatin A, 1b)
Affinity DataKi:  880nM ΔG°:  -36.0kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84464(Benzylation of mannostatin A, 1d)
Affinity DataKi:  910nM ΔG°:  -35.9kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84467(Benzylation of mannostatin A, 1g)
Affinity DataKi:  3.22E+3nM ΔG°:  -32.6kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84474(Aminocyclopentitetrol, 2g)
Affinity DataKi:  4.40E+3nM ΔG°:  -31.8kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84470(Aminocyclopentitetrol, 2c)
Affinity DataKi:  6.00E+3nM ΔG°:  -31.0kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84468(Mannostatin analogue, 4b | Meso-aminocyclopentitet...)
Affinity DataKi:  6.60E+3nM ΔG°:  -30.8kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84473(Aminocyclopentitetrol, 2f)
Affinity DataKi:  6.60E+3nM ΔG°:  -30.8kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84472(Aminocyclopentitetrol, 2e)
Affinity DataKi:  7.60E+3nM ΔG°:  -30.4kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84471(Aminocyclopentitetrol, 2d)
Affinity DataKi:  8.10E+3nM ΔG°:  -30.2kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84469(Aminocyclopentitetrol, 2b)
Affinity DataKi:  1.00E+4nM ΔG°:  -29.7kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed
TargetAlpha-mannosidase 2(Human)
University of Georgia

LigandPNGBDBM84468(Mannostatin analogue, 4b | Meso-aminocyclopentitet...)
Affinity DataKi:  5.00E+4nM ΔG°:  -25.5kJ/molepH: 5.6 T: 2°CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2012
Entry Details Article
PubMed