Compile Data Set for Download or QSAR
Report error Found 33 of ph data with Target = 'Aminopeptidase N'
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240828BDBM240828((2R,3S)-3-amino-2-hydroxy-N-((S)-2-(hydroxyamino)-...)
Affinity DataIC50: 1.26E+3nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 23971BDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 2.50E+3nMpH: 7.2Assay Description:Briefly, the assay was performed in 96-well plates in 50 mm PBS, pH 7.2 as the assay buffer, at 37 °C. The APN solution was mixed with compounds at v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241970BDBM241970(L-isoserine-L-tyrosinase-L-leucyl (16l))
Affinity DataIC50: 2.51E+3nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 23971BDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 2.55E+3nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241968BDBM241968(L-isoserine-L-leucyl-L-valine (16i))
Affinity DataIC50: 5.16E+3nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241966BDBM241966(L-isoserine-L-phenylglycine-L-phenylalanine (16g))
Affinity DataIC50: 5.80E+3nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 23971BDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 6.25E+3nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241972BDBM241972(L-isoserine-L-phenylalanine-L-phenylalanine (16n))
Affinity DataIC50: 6.50E+3nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241967BDBM241967(L-isoserine-L-valine-L-leucyl (16h))
Affinity DataIC50: 6.50E+3nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241964BDBM241964(L-isoserine-L-tyrosinase-L-valine (16e))
Affinity DataIC50: 1.15E+4nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241969BDBM241969(L-isoserine-L-phenylglycine-L-leucyl (16k))
Affinity DataIC50: 1.16E+4nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241965BDBM241965(L-isoserine-L-valine-L-valine (16f))
Affinity DataIC50: 1.36E+4nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241971BDBM241971(L-isoserine-L-eucyl-L-tyrosinase (16m))
Affinity DataIC50: 1.75E+4nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241963BDBM241963(L-isoserine-L-valine-L-phenylalanine (16d))
Affinity DataIC50: 3.02E+4nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241960BDBM241960(2-[2-(3-amino-2-hydroxypropanamido)-3-phenylpropan...)
Affinity DataIC50: 3.04E+4nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240829BDBM240829((2R,3S)-3-amino-2-hydroxy-N-((S)-1-(hydroxyamino)-...)
Affinity DataIC50: 4.40E+4nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241962BDBM241962(L-isoserine-L-phenylglycine-L-valine (16c))
Affinity DataIC50: 5.15E+4nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240824BDBM240824((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 5.67E+4nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240825BDBM240825((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 7.70E+4nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240827BDBM240827((2S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanam...)
Affinity DataIC50: 8.29E+4nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 241961BDBM241961(L-isoserine-L-phenylalanine-L-valine (16b))
Affinity DataIC50: 9.40E+4nMpH: 7.2Assay Description:IC50 values against APN were determined as previously described and by using L-Leu-p-nitroanilide as a substrate and microsomal aminopeptidase from P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 198191BDBM198191(N1-hydroxy-N4-(5,5,8,8-tetramethyl-5,6,7,8-tetrahy...)
Affinity DataIC50: 1.00E+5nMpH: 7.2Assay Description:Briefly, the assay was performed in 96-well plates in 50 mm PBS, pH 7.2 as the assay buffer, at 37 °C. The APN solution was mixed with compounds at v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 50061625BDBM50061625(4-[(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthal...)
Affinity DataIC50: 1.00E+5nMpH: 7.2Assay Description:Briefly, the assay was performed in 96-well plates in 50 mm PBS, pH 7.2 as the assay buffer, at 37 °C. The APN solution was mixed with compounds at v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 19149BDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 1.00E+5nMpH: 7.2Assay Description:Briefly, the assay was performed in 96-well plates in 50 mm PBS, pH 7.2 as the assay buffer, at 37 °C. The APN solution was mixed with compounds at v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240823BDBM240823((S)-2-((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpr...)
Affinity DataIC50: 1.05E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240831BDBM240831((2R,3S)-3-amino-2-hydroxy-N-((S)-3-hydroxy-1-(hydr...)
Affinity DataIC50: 1.58E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240830BDBM240830((2R,3S)-3-amino-2-hydroxy-N-((S)-1-(hydroxyamino)-...)
Affinity DataIC50: 1.73E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240816BDBM240816((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 1.98E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240814BDBM240814((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 3.42E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240812BDBM240812((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 3.52E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240832BDBM240832((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 3.63E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240821BDBM240821((S)-2-((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpr...)
Affinity DataIC50: 5.13E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandChemical structure of BindingDB Monomer ID 240820BDBM240820((S)-2-((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpr...)
Affinity DataIC50: 5.90E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed