Compile Data Set for Download or QSAR
Report error Found 26 of ph data with Target = 'Arachidonate 12-lipoxygenase, 12R-type'
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86082BDBM86082(Tetraketone, 19)
Affinity DataIC50: 7.80E+3nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86085BDBM86085(Tetraketone, 22)
Affinity DataIC50: 1.25E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86070BDBM86070(Tetraketone, 3)
Affinity DataIC50: 1.63E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86077BDBM86077(Tetraketone, 11)
Affinity DataIC50: 1.75E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86074BDBM86074(Tetraketone, 8)
Affinity DataIC50: 2.13E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86072BDBM86072(Tetraketone, 6)
Affinity DataIC50: 2.64E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86080BDBM86080(Tetraketone, 15)
Affinity DataIC50: 2.71E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86078BDBM86078(Tetraketone, 12)
Affinity DataIC50: 2.84E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86076BDBM86076(Tetraketone, 10)
Affinity DataIC50: 3.08E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86069BDBM86069(Tetraketone, 2)
Affinity DataIC50: 3.30E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86075BDBM86075(Tetraketone, 9)
Affinity DataIC50: 3.31E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86083BDBM86083(Tetraketone, 20)
Affinity DataIC50: 3.54E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86087BDBM86087(Buddlejoside B, 2)
Affinity DataIC50: 3.97E+4nMpH: 8.0 T: 2°CAssay Description:Lipoxygenase inhibiting activity was measured by slightly modifying the spectrometric method. Lipoxygenase type I-B and linoleic acid were purchased...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86092BDBM86092(Buddlejoside A5, 7)
Affinity DataIC50: 4.04E+4nMpH: 8.0 T: 2°CAssay Description:Lipoxygenase inhibiting activity was measured by slightly modifying the spectrometric method. Lipoxygenase type I-B and linoleic acid were purchased...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86091BDBM86091(Buddlejoside A2, 6)
Affinity DataIC50: 4.19E+4nMpH: 8.0 T: 2°CAssay Description:Lipoxygenase inhibiting activity was measured by slightly modifying the spectrometric method. Lipoxygenase type I-B and linoleic acid were purchased...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86086BDBM86086(Buddlejoside A, 1)
Affinity DataIC50: 4.43E+4nMpH: 8.0 T: 2°CAssay Description:Lipoxygenase inhibiting activity was measured by slightly modifying the spectrometric method. Lipoxygenase type I-B and linoleic acid were purchased...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86090BDBM86090(Beta-gardiol, 5)
Affinity DataIC50: 4.73E+4nMpH: 8.0 T: 2°CAssay Description:Lipoxygenase inhibiting activity was measured by slightly modifying the spectrometric method. Lipoxygenase type I-B and linoleic acid were purchased...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86089BDBM86089(Genipin, 4)
Affinity DataIC50: 4.96E+4nMpH: 8.0 T: 2°CAssay Description:Lipoxygenase inhibiting activity was measured by slightly modifying the spectrometric method. Lipoxygenase type I-B and linoleic acid were purchased...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86084BDBM86084(Tetraketone, 21)
Affinity DataIC50: 5.15E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86088BDBM86088(Buddlejoside C, 3)
Affinity DataIC50: 5.25E+4nMpH: 8.0 T: 2°CAssay Description:Lipoxygenase inhibiting activity was measured by slightly modifying the spectrometric method. Lipoxygenase type I-B and linoleic acid were purchased...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86079BDBM86079(Tetraketone, 14)
Affinity DataIC50: 5.29E+4nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86010BDBM86010(Chalcone, 10)
Affinity DataKi:  5.76E+4nM ΔG°:  -24.2kJ/molepH: 8.0 T: 2°CAssay Description:In vitro lipoxygenase inhibition assay, lipoxygenase inhibiting activity was convenintly measured by slightly modifying the spectrometic method devel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86012BDBM86012(Chalcone, 11)
Affinity DataKi:  7.17E+4nM ΔG°:  -23.7kJ/molepH: 8.0 T: 2°CAssay Description:In vitro lipoxygenase inhibition assay, lipoxygenase inhibiting activity was convenintly measured by slightly modifying the spectrometic method devel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86081BDBM86081(Tetraketone, 16)
Affinity DataIC50: 1.91E+5nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86073BDBM86073(Tetraketone, 7)
Affinity DataIC50: 1.96E+5nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed
TargetArachidonate 12-lipoxygenase, 12R-type(Human)
Pharmaceutical Research Centre

LigandChemical structure of BindingDB Monomer ID 86071BDBM86071(Tetraketone, 4)
Affinity DataIC50: 1.98E+5nMpH: 8.0 T: 2°CAssay Description:In vitro liposygenase inhibition assay activity was measured by modifying the spectrophotometric method developed by Tappel. The compound was prepar...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2012
Entry Details Article
PubMed