Compile Data Set for Download or QSAR
Report error Found 8 of ph data with Target = 'Cyclin-dependent kinase 5'
TargetCyclin-dependent kinase 5(Human)
Technische UniversitÄT Braunschweig

LigandPNGBDBM84530(Alsterpaullone derivative, 4)
Affinity DataIC50: 23nMpH: 7.5 T: 2°CAssay Description:Kinase activity assay using GSK-3beta, CDK1/cyclin B and CDK5/p25.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Technische UniversitÄT Braunschweig

LigandPNGBDBM84533(BDBM50375663 | Alsterpaullone derivative, 7)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:Kinase activity assay using GSK-3beta, CDK1/cyclin B and CDK5/p25.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Technische UniversitÄT Braunschweig

LigandPNGBDBM7262(NSC 705701 | BDBM84528 | alsterpaullone | 9-Nitrop...)
Affinity DataIC50: 40nMpH: 7.5 T: 2°CAssay Description:Kinase activity assay using GSK-3beta, CDK1/cyclin B and CDK5/p25.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Technische UniversitÄT Braunschweig

LigandPNGBDBM84529(Alsterpaullone derivative, 3)
Affinity DataIC50: 70nMpH: 7.5 T: 2°CAssay Description:Kinase activity assay using GSK-3beta, CDK1/cyclin B and CDK5/p25.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Technische UniversitÄT Braunschweig

LigandPNGBDBM84531(Alsterpaullone derivative, 5)
Affinity DataIC50: 80nMpH: 7.5 T: 2°CAssay Description:Kinase activity assay using GSK-3beta, CDK1/cyclin B and CDK5/p25.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Technische UniversitÄT Braunschweig

LigandPNGBDBM84532(Alsterpaullone derivative, 6)
Affinity DataIC50: 250nMpH: 7.5 T: 2°CAssay Description:Kinase activity assay using GSK-3beta, CDK1/cyclin B and CDK5/p25.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Technische UniversitÄT Braunschweig

LigandPNGBDBM164883(US9067888, 33)
Affinity DataIC50: 1.08E+3nMpH: 7.5Assay Description:In vitro kinase assay analysis may be performed using standard techniques described in the art. These techniques are also used by commercial services...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCyclin-dependent kinase 5(Human)
Technische UniversitÄT Braunschweig

LigandPNGBDBM164884(US9067888, 34)
Affinity DataIC50: 1.34E+3nMpH: 7.5Assay Description:In vitro kinase assay analysis may be performed using standard techniques described in the art. These techniques are also used by commercial services...More data for this Ligand-Target Pair
In DepthDetails
US Patent