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Found 8 of ph data with Target = 'Cyclin-dependent kinase 5'
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Technische UniversitÄT Braunschweig

LigandPNGBDBM84530(Alsterpaullone derivative, 4)
Affinity DataIC50:  23nMpH: 7.5 T: 2°CAssay Description:Kinase activity assay using GSK-3beta, CDK1/cyclin B and CDK5/p25.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Technische UniversitÄT Braunschweig

LigandPNGBDBM84533(Alsterpaullone derivative, 7 | BDBM50375663)
Affinity DataIC50:  30nMpH: 7.5 T: 2°CAssay Description:Kinase activity assay using GSK-3beta, CDK1/cyclin B and CDK5/p25.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Technische UniversitÄT Braunschweig

LigandPNGBDBM7262(14-nitro-8,18-diazatetracyclo[9.7.0.0^{2,7}.0^{12,...)
Affinity DataIC50:  40nMpH: 7.5 T: 2°CAssay Description:Kinase activity assay using GSK-3beta, CDK1/cyclin B and CDK5/p25.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Technische UniversitÄT Braunschweig

LigandPNGBDBM84529(Alsterpaullone derivative, 3)
Affinity DataIC50:  70nMpH: 7.5 T: 2°CAssay Description:Kinase activity assay using GSK-3beta, CDK1/cyclin B and CDK5/p25.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Technische UniversitÄT Braunschweig

LigandPNGBDBM84531(Alsterpaullone derivative, 5)
Affinity DataIC50:  80nMpH: 7.5 T: 2°CAssay Description:Kinase activity assay using GSK-3beta, CDK1/cyclin B and CDK5/p25.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Technische UniversitÄT Braunschweig

LigandPNGBDBM84532(Alsterpaullone derivative, 6)
Affinity DataIC50:  250nMpH: 7.5 T: 2°CAssay Description:Kinase activity assay using GSK-3beta, CDK1/cyclin B and CDK5/p25.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Technische UniversitÄT Braunschweig

LigandPNGBDBM164883(US9067888, 33)
Affinity DataIC50:  1.08E+3nMpH: 7.5Assay Description:In vitro kinase assay analysis may be performed using standard techniques described in the art. These techniques are also used by commercial services...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Technische UniversitÄT Braunschweig

LigandPNGBDBM164884(US9067888, 34)
Affinity DataIC50:  1.34E+3nMpH: 7.5Assay Description:In vitro kinase assay analysis may be performed using standard techniques described in the art. These techniques are also used by commercial services...More data for this Ligand-Target Pair
In DepthDetails US Patent