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Found 157 of ph data with Target = 'Gag-Pol polyprotein [489-587]'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM465((6S)-3-[(4-amino-2-tert-butyl-5-methylphenyl)sulfa...)
Affinity DataKi:  0.0700nMpH: 6.2Assay Description:Binding affinity of the compound towards HIV protease was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078088((S)-3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-pheny...)
Affinity DataKi:  0.0900nMpH: 4.7Assay Description:Inhibitory activity of the compound was evaluated against human immunodeficiency virus type 1(HIV-1) protease at pH 4.7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078088((S)-3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-pheny...)
Affinity DataKi:  0.0900nMpH: 6.2Assay Description:In vitro binding affinity of the compound against HIV protease at pH 6.2 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50216785(CHEMBL61756)
Affinity DataKi: <0.100nMpH: 4.7Assay Description:Inhibitory activity of the compound was evaluated against human immunodeficiency virus type 1(HIV-1) protease at pH 6.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078087((S)-6-[2-(4-Amino-phenyl)-ethyl]-3-(2-tert-butyl-4...)
Affinity DataKi:  0.110nMpH: 6.2Assay Description:In vitro binding affinity of the compound against HIV protease at pH 6.2 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50014015(2-{2-[2-(3-tert-Butoxycarbonylamino-2-hydroxy-4-ph...)
Affinity DataKi:  0.600nMpH: 6.4Assay Description:Inhibition of HIV protease at pH 6.4, 37 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50010497(Acetyl-Ser-Leu-Asn-Phe-[S]-[CH(OH)CH2N]Pro-Ile-Val...)
Affinity DataKi:  0.660nMpH: 6.4Assay Description:Binding affinity against Cysteinyl leukotriene D4 receptor from guinea pig trachea using [3H]LTD4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM396(3-[(4-amino-2-tert-butyl-5-methylphenyl)sulfanyl]-...)
Affinity DataKi:  0.670nMpH: 6.2Assay Description:Binding affinity of the compound towards HIV protease was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50014024(2-(2-{[1-(2-{2-[2-(2-Acetylamino-3-hydroxy-propion...)
Affinity DataKi:  11nMpH: 6.4Assay Description:Inhibitory activity against HIV Protease was measured at pH 6.4 and 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50014020(2-[2-(2-{3-[2-(2-Amino-propionylamino)-propionylam...)
Affinity DataKi:  18nMpH: 6.4Assay Description:Inhibition of HIV protease at pH 6.4, 37 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50014019(2-{2-[(1-{2-[2-(2-Acetylamino-4-methyl-pentanoylam...)
Affinity DataKi:  21nMpH: 6.4Assay Description:Inhibition of HIV protease at pH 6.4, 37 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50421882(CHEMBL2311136)
Affinity DataKi:  21nMpH: 6.4Assay Description:Inhibition of HIV protease at pH 6.4, 37 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50014014(2-{2-[3-(Acetyl-tert-butyl-amino)-4-cyclohexyl-2-h...)
Affinity DataKi:  70nMpH: 6.4Assay Description:Inhibition of HIV protease at pH 6.4, 37 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50014028(2-{[1-(2-{2-[2-(2-Acetylamino-3-hydroxy-propionyla...)
Affinity DataKi:  420nMpH: 6.4Assay Description:Inhibition of HIV protease at pH 6.4, 37 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50014023(2-(2-{3-[2-(2-Acetylamino-3-hydroxy-butyrylamino)-...)
Affinity DataKi:  780nMpH: 6.4Assay Description:Inhibition of HIV protease at pH 6.4, 37 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50014026(2-{[1-(2-{2-[2-(2-Acetylamino-3-hydroxy-propionyla...)
Affinity DataKi:  980nMpH: 6.4Assay Description:Inhibitory activity against HIV Protease was measured at pH 6.4 and 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000902(CHEMBL52494)
Affinity DataKi:  1.06E+3nMpH: 6.4Assay Description:Inhibition of HIV protease at pH 6.4, 37 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000543(CHEMBL417012)
Affinity DataKi:  2.64E+3nMpH: 6.4Assay Description:Inhibition of HIV protease at pH 6.4, 37 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50014018(2-[(1-{2-[2-(2-Acetylamino-4-methyl-pentanoylamino...)
Affinity DataKi:  4.52E+3nMpH: 6.4Assay Description:Inhibition of HIV protease at pH 6.4, 37 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000550(CHEMBL298903)
Affinity DataKi:  8.00E+3nMpH: 6.4Assay Description:Inhibitory activity against HIV Protease was measured at pH 6.4 and 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50014021(2-[(1-{2-[2-(2-Acetylamino-4-methyl-pentanoylamino...)
Affinity DataKi: >1.00E+4nMpH: 6.4Assay Description:Inhibitory activity against HIV Protease was measured at pH 6.4 and 37 degrees CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50281205((3R,5R)-3,5-Dibenzyl-3,4,5-trihydroxy-cyclohexanon...)
Affinity DataKi:  1.00E+4nMpH: 6.0Assay Description:Compound was evaluated for the inhibition of recombinant HIV-1 protease at 37 degrees C and pH of 6.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50014030(2-(2-Acetylamino-3-hydroxy-propionylamino)-pentane...)
Affinity DataKi:  1.30E+4nMpH: 6.4Assay Description:Inhibition of HIV protease at pH 6.4, 37 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50281202((3S,5S)-3,5-Dibenzyl-3,5-bis-hydroxymethyl-1-oxo-t...)
Affinity DataKi:  1.90E+4nMpH: 6.0Assay Description:Compound was evaluated for the inhibition of recombinant HIV-1 protease at 37 degrees C and pH of 6.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50281202((3S,5S)-3,5-Dibenzyl-3,5-bis-hydroxymethyl-1-oxo-t...)
Affinity DataKi:  1.90E+4nMpH: 6.0Assay Description:Compound was evaluated for the inhibition of recombinant HIV-1 protease at 37 degrees C and pH of 6.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000698(CHEMBL49026)
Affinity DataKi:  3.90E+4nMpH: 6.4Assay Description:Inhibition of HIV protease at pH 6.4, 37 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50281207((2S,6S)-2,6-Dibenzyl-2,6-bis-hydroxymethyl-cyclohe...)
Affinity DataKi:  4.80E+4nMpH: 6.0Assay Description:Compound was evaluated for the inhibition of recombinant HIV-1 protease at 37 degrees C and pH of 6.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50281204((3S,5S)-3,5-Dibenzyl-4-hydroxy-3,5-bis-hydroxymeth...)
Affinity DataKi:  6.20E+4nMpH: 6.0Assay Description:Compound was evaluated for the inhibition of recombinant HIV-1 protease at 37 degrees C and pH of 6.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50281206((2S,6S)-2,6-Dibenzyl-2,6-bis-hydroxymethyl-cyclohe...)
Affinity DataKi:  8.30E+5nMpH: 6.0Assay Description:Compound was evaluated for the inhibition of recombinant HIV-1 protease at 37 degrees C and pH of 6.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50281203((2S,6S)-2,6-Dibenzyl-cyclohexane-1,4-diol | CHEMBL...)
Affinity DataKi: >2.00E+6nMpH: 6.0Assay Description:Compound was evaluated for the inhibition of recombinant HIV-1 protease at 37 degrees C and pH of 6.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50281208((1S,3S)-1,3-Dibenzyl-cyclohexane-1,2,3-triol | CHE...)
Affinity DataKi: >2.00E+6nMpH: 6.0Assay Description:Compound was evaluated for the inhibition of recombinant HIV-1 protease at 37 degrees C and pH of 6.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078088((S)-3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-pheny...)
Affinity DataIC50:  1nMpH: 6.2Assay Description:Inhibitory activity of the compound was evaluated against human immunodeficiency virus type 1(HIV-1) protease at pH 6.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50216785(CHEMBL61756)
Affinity DataIC50: <1nMpH: 6.2Assay Description:Inhibitory concentration against human immunodeficiency virus type 1(HIV-1) protease at pH 4.7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50289065(5-[4-Hydroxy-5-(2-isopropyl-phenylsulfanyl)-6-oxo-...)
Affinity DataIC50:  1.80nMpH: 4.7Assay Description:In vitro inhibitory activity against purified HIV-1 protease at a pH of 4.7 and a final enzyme concentration of 0.45-1.1 nMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM396(3-[(4-amino-2-tert-butyl-5-methylphenyl)sulfanyl]-...)
Affinity DataIC50:  2.70nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM420(3-[(4-amino-2-tert-butyl-5-methylphenyl)sulfanyl]-...)
Affinity DataIC50:  3.30nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078086(CHEMBL265095 | N-(5-tert-Butyl-4-{4-hydroxy-6-[2-(...)
Affinity DataIC50:  3.40nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078098(CHEMBL36608 | N-[5-tert-Butyl-4-(4-hydroxy-6-isopr...)
Affinity DataIC50:  3.5nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078095(3-(4-Amino-2-tert-butyl-5-methyl-phenylsulfanyl)-4...)
Affinity DataIC50:  3.80nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078084(3-(4-Amino-2-tert-butyl-5-methyl-phenylsulfanyl)-6...)
Affinity DataIC50:  4.10nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078106(3-(4-Amino-2-tert-butyl-5-methyl-phenylsulfanyl)-6...)
Affinity DataIC50:  4.40nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078093(CHEMBL37597 | N-(5-tert-Butyl-4-{4-hydroxy-6-[2-(4...)
Affinity DataIC50:  5nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078090(CHEMBL432665 | N-(5-tert-Butyl-4-{4-hydroxy-6-[2-(...)
Affinity DataIC50:  5.10nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078103(CHEMBL38154 | N-(5-tert-Butyl-4-{4-hydroxy-6-[2-(4...)
Affinity DataIC50:  5.10nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078109(3-(4-Amino-2-tert-butyl-5-methyl-phenylsulfanyl)-6...)
Affinity DataIC50:  6nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078107(CHEMBL38236 | Pyridine-2-carboxylic acid (5-tert-b...)
Affinity DataIC50:  6.10nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM2183((3-(2-tert-Butyl-4-hydroxy-5-methyl-phenylsulfanyl...)
Affinity DataIC50:  6.5nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50079704(3-(3-tert-Butyl-benzo[b]thiophen-2-ylsulfanyl)-4-h...)
Affinity DataIC50:  7nMpH: 4.7Assay Description:Inhibitory concentration against human immunodeficiency virus type 1(HIV-1) protease at pH 4.7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078108(3-(4-Amino-2-tert-butyl-5-methyl-phenylsulfanyl)-6...)
Affinity DataIC50:  7.5nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50078092(3-(4-Amino-2-tert-butyl-5-methyl-phenylsulfanyl)-4...)
Affinity DataIC50:  7.70nMpH: 6.2Assay Description:In vitro binding affinity against HIV protease at pH 6.2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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