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Found 20 of ph data with Target = 'Methionine aminopeptidase'
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM17871((1S)-1-[5-(benzylsulfanyl)-4H-1,2,4-triazol-3-yl]-...)
Affinity DataIC50:  43.7nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17853(3,5-Pyrazolediamine Inhibitor, 3 | 3-imino-4-[(E)-...)
Affinity DataIC50:  250nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17854(3,5-Pyrazolediamine Inhibitor, 4 | 3-imino-4-[(E)-...)
Affinity DataIC50:  250nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17856(3,5-Pyrazolediamine Inhibitor, 6 | 4-[(E)-2-(3-chl...)
Affinity DataIC50:  550nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17855(3,5-Pyrazolediamine Inhibitor, 5 | 4-[(E)-2-(3-flu...)
Affinity DataIC50:  550nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17857(3,5-Pyrazolediamine Inhibitor, 7 | 4-[(E)-2-(4-flu...)
Affinity DataIC50:  580nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM17870(1,2,4-triazole derivative. | 5-(benzylsulfanyl)-4H...)
Affinity DataIC50:  599nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17858(3,5-Pyrazolediamine Inhibitor, 8 | 4-[(E)-2-(4-chl...)
Affinity DataIC50:  1.25E+3nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17859(3,5-Pyrazolediamine Inhibitor, 9 | 3-imino-4-[(E)-...)
Affinity DataIC50:  1.50E+3nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17863(Amino-Alcohol Inhibitor, 12 | methyl 2-[(2S)-2-[(2...)
Affinity DataIC50:  1.70E+3nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17860(3,5-Pyrazolediamine Inhibitor, 2 | 3-[(E)-2-(5-ami...)
Affinity DataIC50:  1.75E+3nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17861(3,5-Pyrazolediamine Inhibitor, 10 | 3-[(E)-2-(5-am...)
Affinity DataIC50:  2.00E+3nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17864(Amino-Alcohol Inhibitor, 13 | methyl (2S)-2-[(2S)-...)
Affinity DataIC50:  3.50E+3nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM17869((3S)-3-amino-1-(cyclopropylamino)heptane-2,2-diol ...)
Affinity DataIC50:  7.00E+3nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17865(Amino-Alcohol Inhibitor, 14 | methyl (2S)-2-[(2S)-...)
Affinity DataIC50:  1.20E+4nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM17868((2S)-2-amino-4-(methylsulfanyl)-1-(pyridin-2-yl)bu...)
Affinity DataIC50:  1.60E+4nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM17867((2S)-2-amino-4-(methylsulfanyl)-1-(1,3-thiazol-2-y...)
Affinity DataIC50:  1.90E+4nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17862(({4-[(E)-2-(5-amino-3-imino-3H-pyrazol-4-yl)diazen...)
Affinity DataIC50:  2.00E+4nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
The Procter & Gamble Pharmaceuticals

LigandPNGBDBM17866(Amino-Alcohol Inhibitor, 15 | methyl (2S)-2-[(2S)-...)
Affinity DataIC50:  2.50E+4nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of a compound toward EcMAP was measured by incubating the compound at various concentrations in the presence of the enzyme an...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM17872(1,2,4-triazole derivative. | 3-(benzylsulfanyl)-4-...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed