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Found 20 of affinity data with PDB=1UGF
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of human CA2 incubated for 15 mins prior to testing by stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.50E+6nM ΔG°:  -15.8kJ/molepH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of human CA2 incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 assessed as inhibition of CO2 hydration incubated for 15 mins prior to testing by stopped flow C...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of human carbonic anhydrase 2 by Lineweaver-Burk curvesMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.50E+6nMpH: 7.5Assay Description:Inhibition of human carbonic anhydrase 2 after 15 mins by CO2 hydrase assay at pH 7.5More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of human CA2 after 15 mins by stopped-flow/Co2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of human carbonic anhydrase-2 by CO2 hydration reaction based colorimetric stopped-flow methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 assessed as inhibition of CO2 hydration preincubated for 15 mins by Lineweaver-burk plot methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.51E+6nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.51E+6nMAssay Description:Inhibition of human cytosolic carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.51E+6nMAssay Description:Inhibition of human recombinant wild type CA2 by stopped-flow CO2 hydration methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.51E+6nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.51E+6nMAssay Description:Inhibition of human cytosolic carbonic anhydrase-2 preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.51E+6nMpH: 8.3Assay Description:Inhibition of recombinant human carbonic anhydrase 2 after 15 mins by stopped flow CO2 hydration assay at pH 8.3More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.51E+6nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.51E+6nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.51E+6nMAssay Description:Inhibition of human carbonic anhydrase-2 at 20 degC preincubated for 15 mins by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM26985(2-triaza-1,2-diyne | CHEMBL79455 | CHEMBL89295 | N...)
Affinity DataKi:  1.51E+6nM ΔG°:  -15.8kJ/molepH: 7.5 T: 2°CAssay Description:Inhibition of Helicobacter pylori alpha carbonic anhydrase preincubated for 15 mins by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair