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Found 3 of affinity data with PDB=2L84
TargetCREB-binding protein(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50443249(Ischemin)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50443249(Ischemin)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of p53-CBP bromodomain interaction in human U2OS cells assessed as inhibition of p21 activation incubated overnight followed by doxorubici...More data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
University Of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50158615(Ischemin)
Affinity DataKd:  1.96E+4nMAssay Description:Binding affinity to CBP bromodomain (unknown origin) by fluorescence spectroscopic analysisMore data for this Ligand-Target Pair