Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of affinity data with PDB=2VTA
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Astex

LigandPNGBDBM24627(1H-indazole | Indazole, 5 | Indazole, 6)
Affinity DataIC50:  1.85E+5nMpH: 7.2 T: 2°CAssay Description:CDK2/cyclin A activity was determined using a radiometric assay to measure the incorporation of gamma-phosphate from [gamma-33P]-ATP into histone H1....More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM24627(1H-indazole | Indazole, 5 | Indazole, 6)
Affinity DataIC50:  1.85E+5nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM24627(1H-indazole | Indazole, 5 | Indazole, 6)
Affinity DataIC50:  1.85E+5nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) by radiometric filter binding assayMore data for this Ligand-Target Pair