Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Universit£Tsklinikum Frankfurt
Universit£Tsklinikum Frankfurt
Affinity DataIC50: 9.70E+4nMpH: 7.4 T: 2°CAssay Description:The AlphaScreen Assay (Perkin Elmer) was performed according to the manufacturer's protocol in 384-well microtiter plates. Incubations were performe...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Universit£Tsklinikum Frankfurt
Universit£Tsklinikum Frankfurt
Affinity DataKd: 1.03E+4nMAssay Description:Binding affinity to human PDPK1 Y288G/Q292A mutant expressed in insect cell system assessed as substrate phosphorylation by isothermal titration calo...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Universit£Tsklinikum Frankfurt
Universit£Tsklinikum Frankfurt
Affinity DataKd: 1.03E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair