Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of affinity data with PDB=4LCJ
TargetC-terminal-binding protein 2(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM154571(4-Methylthio 2-oxobutyric acid (MTOB))
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus...More data for this Ligand-Target Pair
TargetC-terminal-binding protein 2(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM154571(4-Methylthio 2-oxobutyric acid (MTOB))
Affinity DataKd:  2.96E+6nMpH: 8.5Assay Description:Purified CtBP2 was dialyzed overnight against 500 mL of 50 mM glycylglycine at pH 8.5, 300 mM NaCl, 1 mM EDTA, and 2 mM TCEP, with or without 1.5 mM ...More data for this Ligand-Target Pair
TargetC-terminal-binding protein 1(Homo sapiens (Human))
University Of Massachusetts Medical School

LigandPNGBDBM154571(4-Methylthio 2-oxobutyric acid (MTOB))
Affinity DataKd:  1.26E+6nMpH: 7.5Assay Description:Purified CtBP2 was dialyzed overnight against 500 mL of 50 mM glycylglycine at pH 8.5, 300 mM NaCl, 1 mM EDTA, and 2 mM TCEP, with or without 1.5 mM ...More data for this Ligand-Target Pair