TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Johannes Gutenberg University
Curated by ChEMBL
Johannes Gutenberg University
Curated by ChEMBL
Affinity DataEC50: 1.28E+5nMAssay Description:Agonist activity at rat recombinant GABAAalpha4beta3gamma2 receptor expressed in HEK293 cells assessed as normalization of GABA-induced current by wh...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Homo sapiens (Human))
Moltech
Curated by ChEMBL
Moltech
Curated by ChEMBL
Affinity DataEC50: 3.24E+5nMAssay Description:Activity at alpha-4-beta-3-gamma-2 GABAA receptor expressed in Xenopus oocytes assessed as inhibition in GABA-induced current by voltage clamp assayMore data for this Ligand-Target Pair