Compile Data Set for Download or QSAR
maximum 50k data
Found 11 of ec50 data for polymerid = 10230,49000507,50000084,50001579,50003028,50003030,50003039,50003041,50003066,50004569
TargetEphrin type-A receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50242740(CHEMBL459850 | N-(3-(7-Amino-1-methyl-2-oxo-1,2-di...)
Affinity DataEC50:  2nMAssay Description:Inhibition of EphA3 by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50242740(CHEMBL459850 | N-(3-(7-Amino-1-methyl-2-oxo-1,2-di...)
Affinity DataEC50:  4nMAssay Description:Inhibition of EphB4 by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 2(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50297824(CHEMBL559058 | N-(2-methyl-5-(3-(4-methyl-1H-imida...)
Affinity DataEC50:  40nMAssay Description:Inhibition of EphB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 2(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50297825(5-(2-methyl-5-(3-(trifluoromethyl)phenylcarbamoyl)...)
Affinity DataEC50:  40nMAssay Description:Inhibition of EphB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 2(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50297825(5-(2-methyl-5-(3-(trifluoromethyl)phenylcarbamoyl)...)
Affinity DataEC50:  100nMAssay Description:Inhibition of ephrinB1-induced autophosphorylation of EphB2 expressed in human U87 cells after 1 hr by western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50553180(CHEMBL4792853)
Affinity DataEC50:  360nMAssay Description:Inhibition of full-length human EPHB4 expressed in MEF cells assessed as autophosphorylation by sandwitch-ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM482158(BDBM50242742 | TAE684)
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of EphB4 by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-A receptor 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM482158(BDBM50242742 | TAE684)
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of EphA3 by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50553181(CHEMBL4784484)
Affinity DataEC50:  1.10E+3nMAssay Description:Inhibition of full-length human EPHB4 expressed in MEF cells assessed as autophosphorylation by sandwitch-ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEphrin type-A receptor 2(Homo sapiens (Human))
University Of California Riverside

Curated by ChEMBL
LigandPNGBDBM50588608(CHEMBL5192123)
Affinity DataEC50:  1.60E+3nMAssay Description:Antagonist activity at EPHA2 in human BXPC-3 cells assessed as inhibition of ephrinA1-Fc induced degradation pretreated for 20 mins followed by ephri...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEphrin type-A receptor 7(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50551644(CHEMBL4745937)
Affinity DataEC50:  3.26E+3nMAssay Description:Inhibition of human EPHA7 incubated for 30 mins by Kinobead based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed