TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.00350nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.200nMAssay Description:Agonist activity at human V1B receptor expressed in HEK293 cells assessed as intracellular calcium level measured at 3 secs interval for 5 mins by fu...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.240nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.5nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.800nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed CHO cells assessed as induction of phospholipase C activity after 15 mins by inositol ph...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 1.70nMAssay Description:Binding affinity to human vasopressin V1b receptor expressed CHO cells after 1 hr by spectrofluorimetry analysisMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 2.48nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed CHO cells assessed as induction of phospholipase C activity after 15 mins by inositol ph...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 4.30nMAssay Description:Agonist activity at human vasopressin V1b expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 4.80nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 6.93nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed CHO cells assessed as induction of phospholipase C activity after 15 mins by inositol ph...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 7.5nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 7.70nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 8nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 8.70nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: >10nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: >10nMAssay Description:Agonist activity at human vasopressin V1b expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: >10nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: >10nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: >10nMAssay Description:Agonist activity at human vasopressin V1b expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at human vasopressin V1b expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at recombinant human V1B receptor expressed in HEK293 cells measured after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 18nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 21nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 24nMAssay Description:Agonist activity at recombinant human V1B receptor expressed in HEK293 cells measured after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Agonist activity at human V1b receptor expressed in HEK293FT cells incubated for 30 mins by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 31nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 32nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed in CHO cells assessed as increase in intracellular calcium flux measured for 5 mins by F...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 37nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 38nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 39nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 39nMAssay Description:Agonist activity at human V1b receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at recombinant human V1B receptor expressed in HEK293 cells measured after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 44nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 45nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 46nMAssay Description:Agonist activity at recombinant human V1B receptor expressed in HEK293 cells measured after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 46nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair