Compile Data Set for Download or QSAR
maximum 50k data
Found 83 of ec50 data for polymerid = 2287,50004917,50007028
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204018(CHEMBL3923877)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at rat GPR40 expressed in HEK293 cells assessed as increase in intracellular Ca2+ flux by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168191(US9688642, 2)
Affinity DataEC50:  8nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204019(CHEMBL3927863)
Affinity DataEC50:  10nMAssay Description:Agonist activity at rat GPR40 expressed in HEK293 cells assessed as increase in intracellular Ca2+ flux by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168152(US9688642, 5)
Affinity DataEC50:  11nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50085568(CHEMBL3427712)
Affinity DataEC50:  11nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells assessed as increase in intracellular calcium level after 60 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168173(US9688642, 4)
Affinity DataEC50:  12nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168196(US9688642, 47)
Affinity DataEC50:  14nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50019087(CHEMBL3288348)
Affinity DataEC50:  16nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168166(US9688642, 6)
Affinity DataEC50:  16nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168184(US9688642, 15 | US9688642, 30)
Affinity DataEC50:  18nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168193(US9688642, 9)
Affinity DataEC50:  18nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50339489(3-{4-[(2',6'-Dimethylbiphenyl-3-yl)methoxy]phenyl}...)
Affinity DataEC50:  18nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168159(US9688642, 12)
Affinity DataEC50:  22nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50362690(AMG-837 | CHEMBL1829173)
Affinity DataEC50:  23nMAssay Description:Agonist activity at rat GPR40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168182(US9688642, 14)
Affinity DataEC50:  24nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168190(US9688642, 11)
Affinity DataEC50:  26nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168164(US9688642, 17)
Affinity DataEC50:  28nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168174(US9688642, 7)
Affinity DataEC50:  28nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Macaca fascicularis)
Amgen

Curated by ChEMBL
LigandPNGBDBM50019939(CHEMBL3287569)
Affinity DataEC50:  29nMAssay Description:Agonist activity at cynomolgus monkey GPR40 in presence of 0.01% human serum albumin relative to AMG 837More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168170(US9688642, 3)
Affinity DataEC50:  30nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168199(US9688642, 42)
Affinity DataEC50:  30nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168162(US9688642, 10)
Affinity DataEC50:  31nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168171(US9688642, 1)
Affinity DataEC50:  32nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168175(US9688642, 13)
Affinity DataEC50:  35nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168194(US9688642, 16)
Affinity DataEC50:  37nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50019083(CHEMBL3288344)
Affinity DataEC50:  38nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168157(US9688642, 27)
Affinity DataEC50:  41nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168160(US9688642, 25)
Affinity DataEC50:  42nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168179(US9688642, 22)
Affinity DataEC50:  43nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168177(US9688642, 8)
Affinity DataEC50:  48nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168153(US9688642, 23)
Affinity DataEC50:  54nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168158(US9688642, 28)
Affinity DataEC50:  56nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168167(US9688642, 19)
Affinity DataEC50:  60nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168172(US9688642, 21)
Affinity DataEC50:  61nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168198(US9688642, 44)
Affinity DataEC50:  64nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168155(US9688642, 43)
Affinity DataEC50:  68nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168188(US9688642, 29)
Affinity DataEC50:  72nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50433707(CHEMBL2381282)
Affinity DataEC50:  77nMAssay Description:Agonist activity at GPR40 in rat INS-1 cells assessed as glucose-stimulated insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50019111(CHEMBL3288363)
Affinity DataEC50:  78nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50019110(CHEMBL3288362)
Affinity DataEC50:  79nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168183(US9688642, 31)
Affinity DataEC50:  84nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168169(US9688642, 20)
Affinity DataEC50:  84nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168168(US9688642, 18)
Affinity DataEC50:  86nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50386790(CHEMBL1829174 | CHEMBL2047159 | TAK-875)
Affinity DataEC50:  93nMAssay Description:Agonist activity at GPR40 in rat INS-1 cells assessed as glucose-stimulated insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50019105(CHEMBL3288357)
Affinity DataEC50:  96nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168180(US9688642, 34)
Affinity DataEC50:  98nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM22496(3-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  99nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168154(US9688642, 33)
Affinity DataEC50:  103nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168181(US9688642, 39)
Affinity DataEC50:  104nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM168163(US9688642, 32)
Affinity DataEC50:  106nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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