Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ec50 data for polymerid = 49001044
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Florida Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50024458(5-oxo-ETE | CHEMBL18028 | ETE-5-Oxo)
Affinity DataEC50:  7nMAssay Description:Agonist activity at 5-oxo-ETE receptor in human neutrophils assessed as stimulation of ca2+ mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Florida Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50338299(15-hydroxy-5-oxo-eicosa-6(E),8(Z),11(Z),13(E)tetra...)
Affinity DataEC50:  56nMAssay Description:Agonist activity at 5-oxo-ETE receptor in human neutrophils assessed as stimulation of ca2+ mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Florida Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50024458(5-oxo-ETE | CHEMBL18028 | ETE-5-Oxo)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Florida Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50275217(CHEMBL4127146)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Florida Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50027524(5-Oxo-icosa-6,8,11,14-tetraenoic acid methyl ester...)
Affinity DataEC50:  1.54E+3nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Florida Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50275216(CHEMBL4130040)
Affinity DataEC50:  2.08E+3nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Florida Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50275229(CHEMBL4128214)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Florida Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50275215(CHEMBL4128585)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed