Compile Data Set for Download or QSAR
maximum 50k data
Found 192 of ec50 data for polymerid = 50001651,50002243
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112770((+/-) Propane-2-sulfonic acid [2-(4-iodo-phenyl)-c...)
Affinity DataEC50:  22.6nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112770((+/-) Propane-2-sulfonic acid [2-(4-iodo-phenyl)-c...)
Affinity DataEC50:  22.6nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191952(4-cyano-3-(2'-cyano-biphenyl-4-yl)-5-ethyl-1-methy...)
Affinity DataEC50:  53nMAssay Description:Activity at human recombinant iGluR4 flop expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191952(4-cyano-3-(2'-cyano-biphenyl-4-yl)-5-ethyl-1-methy...)
Affinity DataEC50:  56nMAssay Description:Activity at human recombinant iGluR4 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112771((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  68nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112771((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  68nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191961(4-cyano-5-ethyl-1-methyl-3-(2'-methylsulfanyl-biph...)
Affinity DataEC50:  77nMAssay Description:Activity at human recombinant iGluR4 flop expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191948(4-cyano-5-ethyl-3-(2'-fluoro-biphenyl-4-yl)-1-meth...)
Affinity DataEC50:  80nMAssay Description:Activity at human recombinant iGluR4 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112776((+/-) Propane-2-sulfonic acid [2-(4-iodo-phenyl)-c...)
Affinity DataEC50:  93.1nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112776((+/-) Propane-2-sulfonic acid [2-(4-iodo-phenyl)-c...)
Affinity DataEC50:  93.1nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191961(4-cyano-5-ethyl-1-methyl-3-(2'-methylsulfanyl-biph...)
Affinity DataEC50:  105nMAssay Description:Activity at human recombinant iGluR4 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50094020(CHEMBL136801 | Propane-2-sulfonic acid [2-(4'-amin...)
Affinity DataEC50:  130nMAssay Description:Tested for potentiation towards human iGluR4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112778((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  130nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112778((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  130nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191957(4-cyano-3-(2'-ethoxy-biphenyl-4-yl)-5-ethyl-1-meth...)
Affinity DataEC50:  146nMAssay Description:Activity at human recombinant iGluR4 flop expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50330415((R)-N-(2-(4'-(2-(methylsulfonamido)ethyl)biphenyl-...)
Affinity DataEC50:  150nMAssay Description:Inhibition of GluR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191954(3-(2'-chloro-biphenyl-4-yl)-4-cyano-5-ethyl-1-meth...)
Affinity DataEC50:  157nMAssay Description:Activity at human recombinant iGluR4 flop expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191957(4-cyano-3-(2'-ethoxy-biphenyl-4-yl)-5-ethyl-1-meth...)
Affinity DataEC50:  158nMAssay Description:Activity at human recombinant iGluR4 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50192216(3-(4-tert-butylphenyl)-4-cyano-5-ethylthiophene-2-...)
Affinity DataEC50:  183nMAssay Description:Activity against human GLUR4 flip expressed in HEK293 cells assesed as glutamate-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191948(4-cyano-5-ethyl-3-(2'-fluoro-biphenyl-4-yl)-1-meth...)
Affinity DataEC50:  185nMAssay Description:Activity at human recombinant iGluR4 flop expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112779((+/-) Propane-2-sulfonic acid [2-(4-nitro-phenyl)-...)
Affinity DataEC50:  190nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191955(3-biphenyl-4-yl-4-cyano-5-ethyl-1-methyl-1H-pyrrol...)
Affinity DataEC50:  213nMAssay Description:Activity at human recombinant iGluR4 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191959(3-(4-tert-butylphenyl)-4-cyano-5-(methylthio)thiop...)
Affinity DataEC50:  214nMAssay Description:Activity at human recombinant iGluR4 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191959(3-(4-tert-butylphenyl)-4-cyano-5-(methylthio)thiop...)
Affinity DataEC50:  214nMAssay Description:Activity against human GLUR4 flip expressed in HEK293 cells assesed as glutamate-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191949(4-cyano-5-ethyl-3-(3'-fluoro-biphenyl-4-yl)-1-meth...)
Affinity DataEC50:  223nMAssay Description:Activity at human recombinant iGluR4 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191954(3-(2'-chloro-biphenyl-4-yl)-4-cyano-5-ethyl-1-meth...)
Affinity DataEC50:  225nMAssay Description:Activity at human recombinant iGluR4 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112770((+/-) Propane-2-sulfonic acid [2-(4-iodo-phenyl)-c...)
Affinity DataEC50:  230nMAssay Description:Inhibition of GluR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191951(4-cyano-5-ethyl-3-(4'-fluoro-biphenyl-4-yl)-1-meth...)
Affinity DataEC50:  242nMAssay Description:Activity at human recombinant iGluR4 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112775((+/-) Propane-2-sulfonic acid [2-(4-chloro-phenyl)...)
Affinity DataEC50:  247nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50094034(CHEMBL343972 | Propane-2-sulfonic acid [2-(4'-form...)
Affinity DataEC50:  250nMAssay Description:Tested for potentiation towards human iGluR4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50094016(CHEMBL343571 | Propane-2-sulfonic acid [2-(4'-meth...)
Affinity DataEC50:  270nMAssay Description:Tested for potentiation towards human iGluR4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50192221(3-(4-tert-butylphenyl)-4-cyano-5-(trifluoromethyl)...)
Affinity DataEC50:  273nMAssay Description:Activity against human GLUR4 flip expressed in HEK293 cells assesed as glutamate-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112772((+/-) Propane-2-sulfonic acid [2-(3,5-difluoro-phe...)
Affinity DataEC50:  281nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112772((+/-) Propane-2-sulfonic acid [2-(3,5-difluoro-phe...)
Affinity DataEC50:  281nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50094024((+/-) Propane-2-sulfonic acid [2-(4'-cyano-bipheny...)
Affinity DataEC50:  290nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50094024((+/-) Propane-2-sulfonic acid [2-(4'-cyano-bipheny...)
Affinity DataEC50:  290nMAssay Description:Tested for potentiation towards human iGluR4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50094024((+/-) Propane-2-sulfonic acid [2-(4'-cyano-bipheny...)
Affinity DataEC50:  290nMAssay Description:Inhibition of GluR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191969(4-cyano-3-(4'-cyano-biphenyl-4-yl)-5-ethyl-1-methy...)
Affinity DataEC50:  373nMAssay Description:Activity at human recombinant iGluR4 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191958(4-cyano-5-ethyl-3-(2'-methoxy-biphenyl-4-yl)-1-met...)
Affinity DataEC50:  386nMAssay Description:Activity at human recombinant iGluR4 flop expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191962(3-biphenyl-4-yl-4-cyano-1-methyl-5-methylsulfanyl-...)
Affinity DataEC50:  394nMAssay Description:Activity against human GLUR4 flip expressed in HEK293 cells assesed as glutamate-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50191962(3-biphenyl-4-yl-4-cyano-1-methyl-5-methylsulfanyl-...)
Affinity DataEC50:  394nMAssay Description:Activity at human recombinant iGluR4 flip expressed in HEK293 cells measured as change in intracellular calcium ion concentration in presence of glut...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112781((R,R) Propane-2-sulfonic acid [2-(4-cyano-phenyl)-...)
Affinity DataEC50:  403nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50094024((+/-) Propane-2-sulfonic acid [2-(4'-cyano-bipheny...)
Affinity DataEC50:  420nMAssay Description:Activity against human GLUR4 flip expressed in HEK293 cells assesed as glutamate-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112777((+/-) Propane-2-sulfonic acid (2-p-tolyl-cyclopent...)
Affinity DataEC50:  434nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50192214(3-(4-tert-butylphenyl)-4-cyano-5-(ethylthio)thioph...)
Affinity DataEC50:  440nMAssay Description:Activity against human GLUR4 flip expressed in HEK293 cells assesed as glutamate-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50192222(3-(4-tert-butylphenyl)-4-cyano-5-(dimethylamino)th...)
Affinity DataEC50:  474nMAssay Description:Activity against human GLUR4 flip expressed in HEK293 cells assesed as glutamate-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50192221(3-(4-tert-butylphenyl)-4-cyano-5-(trifluoromethyl)...)
Affinity DataEC50:  488nMAssay Description:Activity against human GLUR4 flop expressed in HEK293 cells assesed as glutamate-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50192223(3-(4-tert-butylphenyl)-4-cyano-5-(methylsulfinyl)t...)
Affinity DataEC50:  489nMAssay Description:Activity against human GLUR4 flip expressed in HEK293 cells assesed as glutamate-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50102263(CHEMBL105076 | N-{4-[1-Methyl-2-(propane-2-sulfony...)
Affinity DataEC50:  520nMAssay Description:Inhibition of GluR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112771((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  520nMAssay Description:Inhibition of GluR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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