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Found 4 of ec50 data for polymerid = 50006140
TargetTopoisomerase I subunit B(Leishmania major)
University Of Puerto Rico

Curated by ChEMBL
LigandPNGBDBM50008923((S)-4-ethyl-4-hydroxy-1,12-dihydro-4H-2-oxa-6,12a-...)
Affinity DataEC50:  670nMAssay Description:Inhibition of Leishmania donovani topoisomerase 1B-mediated relaxation of supercoiled pSK DNA after 30 mins by ethidium bromide staining based agaros...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTopoisomerase I subunit B(Leishmania major)
University Of Puerto Rico

Curated by ChEMBL
LigandPNGBDBM50392269(CHEMBL2153502)
Affinity DataEC50:  5.30E+3nMAssay Description:Inhibition of Leishmania donovani topoisomerase 1B-mediated relaxation of supercoiled pSK DNA after 30 mins by ethidium bromide staining based agaros...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTopoisomerase I subunit B(Leishmania major)
University Of Puerto Rico

Curated by ChEMBL
LigandPNGBDBM50329257(2-Hexadecynoic acid | CHEMBL1269411)
Affinity DataEC50:  2.87E+4nMAssay Description:Inhibition of Leishmania donovani topoisomerase 1B-mediated relaxation of supercoiled pSK DNA after 30 mins by ethidium bromide staining based agaros...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTopoisomerase I subunit B(Leishmania major)
University Of Puerto Rico

Curated by ChEMBL
LigandPNGBDBM50392268(CHEMBL2153501)
Affinity DataEC50:  6.78E+4nMAssay Description:Inhibition of Leishmania donovani topoisomerase 1B-mediated relaxation of supercoiled pSK DNA after 30 mins by ethidium bromide staining based agaros...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed