TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 7.20nMAssay Description:Inhibition of human LDH5 using pyruvate as substrate after 10 minsMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 8.90nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 70nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 90nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 250nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 340nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 390nMAssay Description:Inhibition of human LDH5 using pyruvate as substrate after 10 minsMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 670nMAssay Description:Inhibition of human LDHA using NADH and pyruvate by microplate reader based assayMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 670nMAssay Description:Inhibition of human LDH5 using pyruvate as substrate after 10 minsMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 680nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Inhibition of His-tagged human LDHA incubated for 10 mins using NADH and pyruvate by microplate reader based assayMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 890nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 1.26E+3nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 1.60E+3nMAssay Description:Inhibition of human liver LDHA using sodium pyruvate as substrate after 5 mins in presence of NAPDH and EDTA by diaphorase/resazurin based fluorescen...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 2.14E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 2.56E+3nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 2.90E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 3.03E+3nMAssay Description:Inhibition of human LDHA using NADH and pyruvate by microplate reader based assayMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 3.26E+3nMAssay Description:Inhibition of human LDHA using NADH and pyruvate by microplate reader based assayMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 3.30E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 3.40E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 3.53E+3nMAssay Description:Inhibition of human liver LDHA using sodium pyruvate as substrate after 5 mins in presence of NAPDH and EDTA by diaphorase/resazurin based fluorescen...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 3.70E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 4.10E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 4.58E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 5.60E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 5.70E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 6.40E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 7.50E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 7.80E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 8.18E+3nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 9.70E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 1.24E+4nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human liver LDHA using sodium pyruvate as substrate after 5 mins in presence of NAPDH and EDTA by diaphorase/resazurin based fluorescen...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 1.72E+5nMAssay Description:Binding affinity to human N-terminal His6-tagged human LDH-5 expressed in Escherichia coli Rosetta (DE3) assessed as induction of protein disruption ...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 1.20E+6nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair