Compile Data Set for Download or QSAR
maximum 50k data
Found 41 of ec50 data for polymerid = 5049,5051,10077
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM197160(GNE-140 (6))
Affinity DataEC50:  7.20nMAssay Description:Inhibition of human LDH5 using pyruvate as substrate after 10 minsMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM197160(GNE-140 (6))
Affinity DataEC50:  8.90nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50250655(CHEMBL4059985 | US10961200, Compound 189 | US11247...)
Affinity DataEC50:  70nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524651(CHEMBL1559855)
Affinity DataEC50:  90nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50250656(CHEMBL4081890 | US11247971, Cmpd ID 276)
Affinity DataEC50:  170nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50250677(CHEMBL4100845 | US10961200, Compound 52 | US112479...)
Affinity DataEC50:  250nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524659(CHEMBL1436155)
Affinity DataEC50:  270nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524656(CHEMBL4515658)
Affinity DataEC50:  340nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50275214(CHEMBL4126746)
Affinity DataEC50:  390nMAssay Description:Inhibition of human LDH5 using pyruvate as substrate after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50539400(CHEMBL4648371)
Affinity DataEC50:  670nMAssay Description:Inhibition of human LDHA using NADH and pyruvate by microplate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50275213(CHEMBL4126939)
Affinity DataEC50:  670nMAssay Description:Inhibition of human LDH5 using pyruvate as substrate after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524666(CHEMBL1440413)
Affinity DataEC50:  680nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50535762(CHEMBL4563330)
Affinity DataEC50:  700nMAssay Description:Inhibition of His-tagged human LDHA incubated for 10 mins using NADH and pyruvate by microplate reader based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524650(CHEMBL4461387)
Affinity DataEC50:  890nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524655(CHEMBL4450110)
Affinity DataEC50:  1.20E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM197160(GNE-140 (6))
Affinity DataEC50:  1.26E+3nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM86137(LDHA Inhibitor, 33)
Affinity DataEC50:  1.60E+3nMAssay Description:Inhibition of human liver LDHA using sodium pyruvate as substrate after 5 mins in presence of NAPDH and EDTA by diaphorase/resazurin based fluorescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524657(CHEMBL4462982)
Affinity DataEC50:  1.80E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524652(CHEMBL4556559)
Affinity DataEC50:  2.14E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50250648(CHEMBL4080497 | US10961200, Compound 20 | US112479...)
Affinity DataEC50:  2.56E+3nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524668(CHEMBL4445248)
Affinity DataEC50:  2.90E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50539401(CHEMBL4635477)
Affinity DataEC50:  3.03E+3nMAssay Description:Inhibition of human LDHA using NADH and pyruvate by microplate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50539402(CHEMBL4645847)
Affinity DataEC50:  3.26E+3nMAssay Description:Inhibition of human LDHA using NADH and pyruvate by microplate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524667(CHEMBL4441804)
Affinity DataEC50:  3.30E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524658(CHEMBL4583436)
Affinity DataEC50:  3.40E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50250674(CHEMBL4076973 | US10961200, Compound 53 | US112479...)
Affinity DataEC50:  3.53E+3nMAssay Description:Inhibition of human liver LDHA using sodium pyruvate as substrate after 5 mins in presence of NAPDH and EDTA by diaphorase/resazurin based fluorescen...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524670(CHEMBL1611057)
Affinity DataEC50:  3.70E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524664(CHEMBL4441824)
Affinity DataEC50:  4.10E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524663(CHEMBL4475383)
Affinity DataEC50:  4.58E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524669(CHEMBL1555353)
Affinity DataEC50:  5.60E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524662(CHEMBL4454634)
Affinity DataEC50:  5.70E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524661(CHEMBL4515017)
Affinity DataEC50:  6.40E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524653(CHEMBL4577089)
Affinity DataEC50:  7.50E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524654(CHEMBL4476280)
Affinity DataEC50:  7.80E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50103568(CHEMBL3335794)
Affinity DataEC50:  8.18E+3nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524665(CHEMBL1888862)
Affinity DataEC50:  9.70E+3nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50524660(CHEMBL1554905)
Affinity DataEC50:  1.24E+4nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50250685(CHEMBL1479261 | US10961200, Compound 62 | US112479...)
Affinity DataEC50: >1.00E+5nMAssay Description:Stabilization of LDHA in human A673 cell lysate preincubated for 20 mins followed by incubation at 70 degreeC for 10 mins by cellular thermal shift a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50250652(CHEMBL4101800 | US10961200, Compound 42 | US112479...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human liver LDHA using sodium pyruvate as substrate after 5 mins in presence of NAPDH and EDTA by diaphorase/resazurin based fluorescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50527803(CHEMBL4557180)
Affinity DataEC50:  1.72E+5nMAssay Description:Binding affinity to human N-terminal His6-tagged human LDH-5 expressed in Escherichia coli Rosetta (DE3) assessed as induction of protein disruption ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50144744(Sodium Oxamate)
Affinity DataEC50:  1.20E+6nMAssay Description:Inhibition of recombinant human full-length N-terminal His-tagged LDHA (1 to 332 residues) expressed in Escherichia coli using sodium pyruvate as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed