Compile Data Set for Download or QSAR
maximum 50k data
Found 959 of ec50 data for polymerid = 5779,5893,50004101,50004885
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM109573(US8604061, 369)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM50158488(CHEMBL3781675)
Affinity DataEC50:  1nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM109570(US8604061, 364)
Affinity DataEC50:  1nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM96729(2-[5-[[anilino(oxo)methyl]amino]-1,3,4-thiadiazol-...)
Affinity DataEC50: >1.5nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM96777(MLS001181838 | N-[4-(phenylcarbamoylamino)phenyl]a...)
Affinity DataEC50: >1.5nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50022723((+)-(S)-amphetamine | (+)-alpha-methylphenethylami...)
Affinity DataEC50:  2nMAssay Description:Activation of mouse TAAR1 expressed in human HEK293 cells assessed as accumulation of cAMP after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM50181823(CHEMBL425035 | O-phenyl-3-iodotyramine)
Affinity DataEC50:  2.40nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM50181812(CHEMBL382580 | O-(p-fluoro)phenyl-3-iodotyramine)
Affinity DataEC50:  2.70nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50158431(CHEMBL3779993)
Affinity DataEC50:  3nMAssay Description:Agonist activity at mouse TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50581608(CHEMBL5082760)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at recombinant human TAAR1 expressed in CHO-K1 cells assessed as increase in intracellular cAMP incubated for 30 mins by HTRF analys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50022723((+)-(S)-amphetamine | (+)-alpha-methylphenethylami...)
Affinity DataEC50:  4nMAssay Description:Activation of mouse TAAR1 transmembrane domain 6 Thr268(6.55)Met mutant expressed in HEK293 cells assessed as stimulation of cAMP production after 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM106582(CHEMBL2206890 | US8586617, 23)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at human TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM106574(CHEMBL2206404 | US8586617, 7)
Affinity DataEC50:  6.80nMAssay Description:Agonist activity at human TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM106574(CHEMBL2206404 | US8586617, 7)
Affinity DataEC50:  7.30nMAssay Description:Agonist activity at rat TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM109388(US8604061, 91)
Affinity DataEC50:  8nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50227513(2-(thiophen-2-yl)ethanamine | CHEMBL252803)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity at recombinant human TAAR1 expressed in CHO-K1 cells assessed as increase in intracellular cAMP incubated for 30 mins by HTRF analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM122294(US8729113, 1)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM106582(CHEMBL2206890 | US8586617, 23)
Affinity DataEC50:  10nMAssay Description:Agonist activity at mouse TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50158488(CHEMBL3781675)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50181798(CHEMBL202335 | N-methyl-O-(p-trifluoromethyl)benzy...)
Affinity DataEC50:  12nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM109573(US8604061, 369)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM50022723((+)-(S)-amphetamine | (+)-alpha-methylphenethylami...)
Affinity DataEC50:  14nMAssay Description:Activation of rat TAAR1 transmembrane domain 7 Asn287(7.39)Tyr mutant expressed in HEK293 cells assessed as stimulation of cAMP production after 1 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM50158431(CHEMBL3779993)
Affinity DataEC50:  14nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50158472(CHEMBL3780993)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM10758(14C-phenylethylamine | 2-phenylethan-1-amine | CHE...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at recombinant human TAAR1 expressed in CHO-K1 cells assessed as increase in intracellular cAMP incubated for 30 mins by HTRF analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50158471(CHEMBL3781694)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM109487(US8604061, 231)
Affinity DataEC50:  18nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50359499((S)Methamphetamine | METHAMPHETAMINE)
Affinity DataEC50:  18nMAssay Description:Activation of mouse TAAR1 transmembrane domain 6 Thr268(6.55)Met mutant expressed in HEK293 cells assessed as stimulation of cAMP production after 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM109524(US8604061, 292)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM109488(US8604061, 232)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM50181802(CHEMBL202024 | N-methyl-3-iodothyronamine)
Affinity DataEC50:  18nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM50212671(2-(3-phenoxyphenyl)-2-phenylethylamine hydrochlori...)
Affinity DataEC50:  19nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50181821(CHEMBL202071 | O-(p-trifluoromethyl)benzyl-tyramin...)
Affinity DataEC50:  20.2nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM109455(US8604061, 192)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50181814(CHEMBL201993 | O-(p-nitro)benzyl-tyramine)
Affinity DataEC50:  21.5nMAssay Description:Activity at mouse TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM50359505(CHEMBL1182312)
Affinity DataEC50:  22.4nMAssay Description:Activation of rat TAAR1 expressed in Syrian hamster AV12-664 cells assessed as accumulation of cAMP after 30 mins using cAMP XS EA/CL as substrate by...More data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM106586(CHEMBL2206375 | US8586617, 28)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM109348(US8604061, 4)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM106586(CHEMBL2206375 | US8586617, 28)
Affinity DataEC50:  23nMAssay Description:Agonist activity at mouse TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM96823(7-methyl-N-(2-phenylethyl)-8-(3,4,5-trimethoxyphen...)
Affinity DataEC50:  23.9nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50581616(CHEMBL4555465)
Affinity DataEC50:  25nMAssay Description:Agonist activity at recombinant human TAAR1 expressed in CHO-K1 cells assessed as increase in intracellular cAMP incubated for 30 mins by HTRF analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM106586(CHEMBL2206375 | US8586617, 28)
Affinity DataEC50:  25nMAssay Description:Agonist activity at rat TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM106608(CHEMBL2206388 | US8586617, 113)
Affinity DataEC50:  25nMAssay Description:Agonist activity at rat TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM50212661(2-(1-phenoxynaphthalen-4-yl)ethylamine | CHEMBL229...)
Affinity DataEC50:  26nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM109570(US8604061, 364)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM106582(CHEMBL2206890 | US8586617, 23)
Affinity DataEC50:  27nMAssay Description:Agonist activity at rat TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50158480(CHEMBL3780421)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50158476(CHEMBL3781589)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM109379(US8604061, 80 (S))
Affinity DataEC50:  27nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM106574(CHEMBL2206404 | US8586617, 7)
Affinity DataEC50:  28nMAssay Description:Agonist activity at mouse TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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