Compile Data Set for Download or QSAR
maximum 50k data
Found 39 of ic50 data for polymerid = 255,10319,50000205
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50326056((1S,3aR,6aS)-2-((S)-2-((S)-2-cyclohexyl-2-(pyrazin...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human Pancreatic elastase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50312532(CHEMBL1077010 | molassamide)
Affinity DataIC50:  32nMAssay Description:Inhibition of pig pancreatic elastase preincubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50038879((S)-2-(2-Formyl-pyrrolidine-1-carbonyl)-pyrrolidin...)
Affinity DataIC50:  51.6nMAssay Description:Inhibition of Flavobacterium meningosepticum PEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Bovine)
University Of Helsinki

LigandPNGBDBM65489(MdnA7)
Affinity DataIC50:  1.05E+3nMT: 2°CAssay Description:The inhibition assays were performed in 96-well microtiter plates as follows: 30 uL of the enzyme solution (trypsin [100 ug/mL] or elastase [1.5 U/mL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50269565(CHEMBL500199 | propeptin)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Flavobacterium meningosepticum PEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50269564(5,6,5',6'-tetrahydroxy[3,3']bibenzofuranyl-2,2'-di...)
Affinity DataIC50:  1.14E+3nMAssay Description:Inhibition of Flavobacterium meningosepticum PEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50269567(CHEMBL515528 | Kynapcin-12)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of Flavobacterium meningosepticum PEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50269566(CHEMBL458248 | polyozellin)
Affinity DataIC50:  2.72E+3nMAssay Description:Inhibition of Flavobacterium meningosepticum PEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50326055((1R,21S,24S)-21-tert-Butyl-N-((1R,2R)-1-{[(cyclopr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human Pancreatic elastase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM12311((1R,5S)-N-[3-Amino-1-(cyclobutylmethyl)-2,3-dioxop...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human Pancreatic elastase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50302107(CHEMBL567893 | Grassystatin A)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of porcine pancreatic elastase after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50310584(CHEMBL1078049 | N-(5-Chloro-pyridin-2-yl)-2-(4-{N-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237204(Esculin laurate)
Affinity DataIC50:  2.00E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Bovine)
University Of Helsinki

LigandPNGBDBM65491(MdnA8)
Affinity DataIC50:  2.19E+4nMT: 2°CAssay Description:The inhibition assays were performed in 96-well microtiter plates as follows: 30 uL of the enzyme solution (trypsin [100 ug/mL] or elastase [1.5 U/mL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237205(Esculin myristate)
Affinity DataIC50:  2.50E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237206(Esculin palmitate)
Affinity DataIC50:  3.00E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  5.00E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237207(Esculin stearate)
Affinity DataIC50:  6.00E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237198(Phloridzin)
Affinity DataIC50:  1.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237184(Rutin)
Affinity DataIC50:  1.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237203(Esculin)
Affinity DataIC50:  1.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237201(Phloridzin palmitate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237202(Phloridzin stearate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237199(Phloridzin laurate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237197(Rutin erucate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237208(4-Guanidinobenzoate)
Affinity DataIC50:  5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237196(Rutin arachidonate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237195(Rutin linolenate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237194(Rutin linoleate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237193(Rutin oleate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237192(Rutin stearate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237191(Rutin palmitate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237190(Rutin myristate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237189(Rutin laurate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237186(Rutin caproate | Rutin capronate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237187(Rutin caprylate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237186(Rutin caproate | Rutin capronate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237185(Rutin butyrate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237200(Phloridzin myristate)
Affinity DataIC50: >5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed