Compile Data Set for Download or QSAR
maximum 50k data
Found 88 of ic50 data for polymerid = 3737,49000030,49000033
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50240412(3-(4-{7-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexen...)
Affinity DataIC50:  99nMAssay Description:Binding affinity to 5HT1E receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50240412(3-(4-{7-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexen...)
Affinity DataIC50:  99nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1E receptor subtypeMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50285314(3-(4-{8-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexen...)
Affinity DataIC50:  392nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1E receptor subtypeMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31044(1-Ethyl-6-methyl-3-thiophen-2-yl-1H-pyrimido[5,4-e...)
Affinity DataIC50:  629nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31041(3-Bromo-4-chloro-7-diethylamino-chromen-2-one | 3-...)
Affinity DataIC50:  999nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50285315(3-(4-{2-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexen...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1E receptor subtypeMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50285317(3-(4-{3-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexen...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1E receptor subtypeMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50285313(3-(4-{10-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexe...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1E receptor subtypeMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50285316(3-(4-{6-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexen...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1E receptor subtypeMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50285318(3-(4-{5-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexen...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1E receptor subtypeMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50285312(3-(4-{4-[4-(5-carbamoyl-1H-3-indolyl)-3-cyclohexen...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1E receptor subtypeMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31072(2-[(1,1-dioxido-1-benzothien-3-yl)thio]-5-phenyl-1...)
Affinity DataIC50:  1.04E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31361(MLS000391019 | N-[3-chloro-4-(difluoromethoxy)phen...)
Affinity DataIC50:  1.25E+3nMpH: 7.4 T: 2°CAssay Description:The CHO cell line was cultured in T-175 flasks at 37 degrees C and 95% relative humidity (RH). The growth media consisted of Dulbecco's Modified ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31347(2-(3,4-dimethoxyphenyl)-N-[3-[5-(3-methylphenyl)-1...)
Affinity DataIC50:  1.76E+3nMpH: 7.4 T: 2°CAssay Description:The CHO cell line was cultured in T-175 flasks at 37 degrees C and 95% relative humidity (RH). The growth media consisted of Dulbecco's Modified ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31053(8-fluoranyl-4-[4-(3-methoxyphenyl)-3-methyl-pipera...)
Affinity DataIC50:  1.82E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31352(2-Cyclopentyl-N-naphthalen-2-yl-2-phenyl-acetamide...)
Affinity DataIC50:  1.85E+3nMpH: 7.4 T: 2°CAssay Description:The CHO cell line was cultured in T-175 flasks at 37 degrees C and 95% relative humidity (RH). The growth media consisted of Dulbecco's Modified ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31054((2E)-3,3,3-trifluoro-2-(4-keto-6-methyl-[1,3]oxath...)
Affinity DataIC50:  1.87E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31068(2-(methylsulfonyl)-4-thien-2-yl-6-(trifluoromethyl...)
Affinity DataIC50:  1.93E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31364((1S,2S)-2-Phenyl-cyclopropanecarboxylic acid [1-[5...)
Affinity DataIC50:  1.96E+3nMpH: 7.4 T: 2°CAssay Description:The CHO cell line was cultured in T-175 flasks at 37 degrees C and 95% relative humidity (RH). The growth media consisted of Dulbecco's Modified ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31042((5-acetamido-4-acetyloxy-2,1,3-benzoxadiazol-7-yl)...)
Affinity DataIC50:  2.10E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31063(2-(methylsulfonyl)-4-phenyl-6-(trifluoromethyl)pyr...)
Affinity DataIC50:  2.13E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31064(4-(2-furanyl)-2-methylsulfonyl-6-(trifluoromethyl)...)
Affinity DataIC50:  2.26E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31082(5,5-dimethyl-2-[(2-methylsulfanylanilino)methylide...)
Affinity DataIC50:  2.36E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31363(MLS000563797 | N-[(R)-[(1R,2R)-2-butylcyclopropyl]...)
Affinity DataIC50:  2.47E+3nMpH: 7.4 T: 2°CAssay Description:The CHO cell line was cultured in T-175 flasks at 37 degrees C and 95% relative humidity (RH). The growth media consisted of Dulbecco's Modified ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31372(3-(2-furanyl)-5-(4-nitrophenyl)-2-phenyl-3,4-dihyd...)
Affinity DataIC50:  2.49E+3nMpH: 7.4 T: 2°CAssay Description:The CHO cell line was cultured in T-175 flasks at 37 degrees C and 95% relative humidity (RH). The growth media consisted of Dulbecco's Modified ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31076(2-[1-(4-methoxyphenyl)tetrazol-5-yl]sulfonyl-1-pip...)
Affinity DataIC50:  2.61E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31083(MLS000107813 | SMR000103777 | [4-(4,7-dimethyl-1,3...)
Affinity DataIC50:  2.62E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31066(3-(1-phenyltetrazol-5-yl)sulfonylpropanenitrile | ...)
Affinity DataIC50:  2.79E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31062(5-methyl-N-(5-quinolinyl)-2-thiophenesulfonamide |...)
Affinity DataIC50:  2.91E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31067(4-(3,4-dimethoxyphenyl)-2-(methylsulfonyl)-6-(trif...)
Affinity DataIC50:  2.91E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31061(4-[1-(4-chlorophenyl)tetrazol-5-yl]sulfanylthieno[...)
Affinity DataIC50:  3.50E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31060(1-cyclopentyl-3-(1-methyl-2-benzimidazolyl)-2-pyrr...)
Affinity DataIC50:  3.64E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31074(MLS000062611 | N-(6-methoxy-8-quinolinyl)-4-methyl...)
Affinity DataIC50:  3.75E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31371(3-(tert-butyl)-N-(4-fluorophenyl)-1-(3-methylbenzy...)
Affinity DataIC50:  3.86E+3nMpH: 7.4 T: 2°CAssay Description:The CHO cell line was cultured in T-175 flasks at 37 degrees C and 95% relative humidity (RH). The growth media consisted of Dulbecco's Modified ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31043(3,6-dioxido-7-(p-tolyl)-4,5-dihydrotriazolo[4,5-e]...)
Affinity DataIC50:  3.91E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31081(7-(hydroxymethyl)-2-(4-phenylphenyl)-4,7a-dihydro-...)
Affinity DataIC50:  4.91E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31071((E)-3-[5-(1-azepanyl)-2-furanyl]-2-(4-fluorophenyl...)
Affinity DataIC50:  5.20E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31362(2-chlorobenzoic acid [2-(3-chloro-4-methyl-anilino...)
Affinity DataIC50:  5.28E+3nMpH: 7.4 T: 2°CAssay Description:The CHO cell line was cultured in T-175 flasks at 37 degrees C and 95% relative humidity (RH). The growth media consisted of Dulbecco's Modified ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31355(2,2-Di-m-tolyl-cyclopropanecarboxylic acid (2-hydr...)
Affinity DataIC50:  5.46E+3nMpH: 7.4 T: 2°CAssay Description:The CHO cell line was cultured in T-175 flasks at 37 degrees C and 95% relative humidity (RH). The growth media consisted of Dulbecco's Modified ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50005835((3-[2-(dimethylamino)ethyl]-1H-indol-5-yl)-N-methy...)
Affinity DataIC50:  5.50E+3nMAssay Description:Compound was evaluated for the affinity at 5-hydroxytryptamine 1E receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31080(1-(2,4-dimethylphenyl)-4-[4-(3-methoxyphenyl)-1-pi...)
Affinity DataIC50:  6.99E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31353(2-Cyclopentyl-2-phenyl-N-p-tolyl-acetamide | 2-cyc...)
Affinity DataIC50:  7.06E+3nMpH: 7.4 T: 2°CAssay Description:The CHO cell line was cultured in T-175 flasks at 37 degrees C and 95% relative humidity (RH). The growth media consisted of Dulbecco's Modified ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31051(4-[4-(3-methoxyphenyl)-3-methyl-1-piperazinyl]-5H-...)
Affinity DataIC50:  8.24E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31046(3-[4,5-dihydro-1H-imidazol-2-ylmethyl-(4-methylphe...)
Affinity DataIC50:  9.22E+3nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31350(1-(4-nitrophenyl)-N-(p-tolyl)cyclopentanecarboxami...)
Affinity DataIC50:  9.48E+3nMpH: 7.4 T: 2°CAssay Description:The CHO cell line was cultured in T-175 flasks at 37 degrees C and 95% relative humidity (RH). The growth media consisted of Dulbecco's Modified ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50304075(3-(5-(4-tert-butylphenyl)-3-((dimethylamino)methyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of 5HT1E receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50060429((R)-2-(4-Fluoro-phenyl)-2-{1-[3-(5-[1,2,4]triazol-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for the displacement of [3H]-5-HT binding to cloned human 5-hydroxytryptamine 1E receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50060437(3-(3-{4-[2-(3-Fluoro-phenyl)-ethyl]-piperazin-1-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was evaluated for the affinity at 5-hydroxytryptamine 1E receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31052(1-[1,1-bis(trifluoromethyl)propyl]-3-[5-(trifluoro...)
Affinity DataIC50:  1.01E+4nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM31046(3-[4,5-dihydro-1H-imidazol-2-ylmethyl-(4-methylphe...)
Affinity DataIC50:  1.08E+4nMpH: 7.4 T: 2°CAssay Description:To measure 5-HT1E activity, a Chinese Hamster Ovary (CHO) cell line was developed at the Scripps Molecular Research Institute Screening center. This ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
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