TargetAmine oxidase [flavin-containing] B(Mus musculus)
R.C. Patel Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
R.C. Patel Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of mouse brain MAO-BMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Mus musculus)
R.C. Patel Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
R.C. Patel Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of mouse brain MAO-BMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.0140nMAssay Description:Inhibitory concentration against Monoamine oxidase B was measured in baboon liver.More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.0170nMAssay Description:Inhibition of human monoamine oxidase BMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 0.0250nMAssay Description:Inhibition of mitochondrial MAO-B in rat liver homogenates using [14C]-phenylethylamine as substrate preincubated for 30 mins by liquid scintillation...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.0480nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.134nMAssay Description:Inhibition of human MAO-B using p-tyramine as substrate after 15 mins by amplex red reagent based assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.227nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus-infected insect cells using p-tyraimne substrateMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.310nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect BT1-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramine up to 15 min...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.318nMAssay Description:Inhibitory concentration against Monoamine oxidase B was measuredMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Inhibition of human MAO-BMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.386nMAssay Description:Inhibition of recombinant human MAOB expressed in baculovirus-infected BTI insect cells using p-tyramine as substrate measured for 45 mins in presenc...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.386nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus-infected insect cells using p-tyraimne substrateMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.389nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Mus musculus)
R.C. Patel Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
R.C. Patel Institute Of Pharmaceutical Education And Research
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of mouse muscle MAO-BMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human microsomal MAO-B expressed in recombinant baculovirus infected insect BTI-TN-5B1-4 cells assessed as reduction in H2O2 production...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:In vitro inhibitory activity against monoamine oxidase B (MAO-B) in rat brain homogenate.More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.407nMAssay Description:Inhibition of human microsomal MAO-B expressed in recombinant baculovirus infected insect BTI-TN-5B1-4 cells assessed as reduction in H2O2 production...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of MAO-B in rat whole brain homogenate in presence of clorgylineMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Stimulation of [35S]GTPcS binding against recombinant human opioid receptor mu 1More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibitory activity against monoamine oxidase B (MAO-B) in rat brain homogenate.More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.586nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus-infected insect cells using p-tyraimne substrateMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.586nMAssay Description:Inhibition of recombinant human MAOB expressed in baculovirus-infected BTI insect cells using p-tyramine as substrate measured for 45 mins in presenc...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.588nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected insect cells assessed as hydrogen peroxide production using p-tyramine as sub...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.589nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:In vitro inhibitory activity against monoamine oxidase B (MAO-B) in rat brain homogenate.More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.612nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus-infected insect cells using p-tyraimne substrateMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.617nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.660nMAssay Description:Inhibition of human recombinant MAOB expressed in insect cells by fluorescence assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.661nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.662nMAssay Description:Inhibition of recombinant human MAOB expressed in baculovirus-infected BTI insect cells using p-tyramine as substrate measured for 45 mins in presenc...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.668nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus-infected insect cells using p-tyraimne substrateMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.670nMAssay Description:Inhibition of human microsomal MAO-B expressed in recombinant baculovirus infected insect BTI-TN-5B1-4 cells assessed as reduction in H2O2 production...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.676nMAssay Description:Inhibition of human microsomal MAO-B expressed in recombinant baculovirus infected insect BTI-TN-5B1-4 cells assessed as reduction in H2O2 production...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.676nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.679nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus-infected insect cells using p-tyraimne substrateMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.679nMAssay Description:Inhibition of recombinant human MAOB expressed in baculovirus-infected BTI insect cells using p-tyramine as substrate measured for 45 mins in presenc...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human recombinant MAO-B using p-tyramine as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr b...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.740nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect BT1-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramine up to 15 min...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.770nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected insect cells assessed as hydrogen peroxide production using p-tyramine as sub...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:In vitro inhibitory activity against monoamine oxidase B (MAO-B) in rat brain homogenate.More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human recombinant MAO-B expressed in insect BT1-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramine up to 15 min...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human recombinant MAO-B using p-tyramine as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr b...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.803nMAssay Description:Inhibition of human recombinant MAOB expressed in BTI cellsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.875nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected insect cells assessed as hydrogen peroxide production using p-tyramine as sub...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.890nMAssay Description:IC50 values for the inhibition of MAO-A and MAO-B were determined using the recombinant human enzymes as enzyme sources, and kynuramine as non-select...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic)
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:In vitro inhibitory activity against monoamine oxidase B (MAO-B) in rat brain homogenate.More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of MAO-B (unknown origin)More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
FacultéS Universitaires Notre-Dame De La Paix
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair