Found 4024 of ic50 data for polymerid = 495,3630,5866,7891,49000449,49000460,49000462,49000463,49000466,49000468,50003096
Affinity DataIC50: >0nMAssay Description:Antagonist required to inhibit Dopamine receptor D2 photoinactivation by 50% with Iodazidoclebopride using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: 0nMAssay Description:Agonist required to inhibit Dopamine receptor D2 photoinactivation by 50% with Iodazidoclebopride using [3H]-SpiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: 0nMAssay Description:Agonist required to inhibit Dopamine receptor D2 photoinactivation by 50% with Iodazidoclebopride using [3H]-SpiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: 0nMAssay Description:Agonist required to inhibit Dopamine receptor D2 photoinactivation by 50% with Iodazidoclebopride using [3H]-SpiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: 0nMAssay Description:Antagonist required to inhibit Dopamine receptor D2 photoinactivation by 50% with Iodazidoclebopride using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: 0nMAssay Description:Agonist required to inhibit Dopamine receptor D2 photoinactivation by 50% with Iodazidoclebopride using [3H]-SpiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: 0nMAssay Description:Antagonist required to inhibit Dopamine receptor D2 photoinactivation by 50% with Iodazidoclebopride using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: 0nMAssay Description:Antagonist required to inhibit Dopamine receptor D2 photoinactivation by 50% with Iodazidoclebopride using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: 0nMAssay Description:Agonist required to inhibit Dopamine receptor D2 photoinactivation by 50% with Iodazidoclebopride using [3H]-SpiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: 0nMAssay Description:Agonist required to inhibit Dopamine receptor D2 photoinactivation by 50% with Iodazidoclebopride using [3H]-SpiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0600nMAssay Description:In vitro inhibition of [3H]-spiroperidol binding to rat Dopamine D2 receptors.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:Displacement of [3H]raclopride from rat dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0710nMAssay Description:Displacement of [3H]raclopride from rat dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0710nMAssay Description:Binding affinity against Dopamine receptor D2 from rat brain corpus striatum membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0750nMAssay Description:In vivo binding affinity of the compound against dopamine (D2) receptor in rat caudate-putamen tissue using [3H]-nemonapride as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0920nMAssay Description:The D2 receptor agonism activity test (The agonism activity of test compounds on D2 receptor expressing human recombinant D2 receptor in HEK293 cells...More data for this Ligand-Target Pair
Affinity DataIC50: 0.123nMAssay Description:Antagonist activity at D2 long receptor (unknown origin) transfected in human HEK293T cells assessed as increase in cAMP accumulation incubated for 2...More data for this Ligand-Target Pair
Affinity DataIC50: 0.124nMAssay Description:Antagonist activity at D2 long receptor (unknown origin) transfected in human HEK293T cells assessed as increase in cAMP accumulation incubated for 2...More data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Antagonist activity at recombinant human D2 receptor expressed in CHOK1 cells assessed as inhibition of quinpirole-induced beta arrestin2 recruitment...More data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Antagonist activity against human D2LR expressed in CHOK1 cells assessed as inhibition of pergolide-induced beta-arrestin translocation by beta-galac...More data for this Ligand-Target Pair
Affinity DataIC50: 0.219nMAssay Description:The D2 receptor agonism activity test (The agonism activity of test compounds on D2 receptor expressing human recombinant D2 receptor in HEK293 cells...More data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:Displacement of [3H]-spiperone from rat striatum D2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.242nMAssay Description:The D2 receptor agonism activity test (The agonism activity of test compounds on D2 receptor expressing human recombinant D2 receptor in HEK293 cells...More data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Displacement of [3H]Spiperone from human recombinant dopamine D2S receptor expressed in CHO cells after 2 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.288nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMT: 2°CAssay Description:Antagonist activity at dopamine D2 receptor (unknown origin) expressed in CHOK1 cells coexpressing Galpha15 assessed as inhibition of agonist-induced...More data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:The D2 receptor agonism activity test (The agonism activity of test compounds on D2 receptor expressing human recombinant D2 receptor in HEK293 cells...More data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Binding affinity against Dopamine receptor D2 from rat brain corpus striatum membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.360nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal dopamine receptor D2 was determined in vitroMore data for this Ligand-Target Pair
Affinity DataIC50: 0.384nMAssay Description:The D2 receptor agonism activity test (The agonism activity of test compounds on D2 receptor expressing human recombinant D2 receptor in HEK293 cells...More data for this Ligand-Target Pair
Affinity DataIC50: 0.480nMAssay Description:Binding affinity to dopamine receptor D2 using a [3H]-spiperone binding assay in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.480nMAssay Description:The D2 receptor agonism activity test (The agonism activity of test compounds on D2 receptor expressing human recombinant D2 receptor in HEK293 cells...More data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Inhibitory concentration required for displacing radioligand [3H]SPI from DA D-2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of binding of radioligand [3H]-spiroperidol to dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]-spiroperidol as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 0.501nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.620nMAssay Description:In vitro inhibitory activity against [3H]raclopride binding to dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataIC50: 0.620nMAssay Description:In vitro inhibition of [3H]-spiperone binding to Dopamine receptor D2 in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.650nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal dopamine receptor D2 was determined in vitroMore data for this Ligand-Target Pair
Affinity DataIC50: 0.672nMAssay Description:The D2 receptor agonism activity test (The agonism activity of test compounds on D2 receptor expressing human recombinant D2 receptor in HEK293 cells...More data for this Ligand-Target Pair
Affinity DataIC50: 0.676nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptor of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at human dopamine D2 short receptor transiently expressed in HEK293 cells assessed as inhibition of beta-arrestin recruitment aft...More data for this Ligand-Target Pair
Affinity DataIC50: 0.740nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.760nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(BOVINE)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 0.770nMAssay Description:Affinity towards Dopamine receptor D2 in membranes from bovine striatum using [3H]-racloprideMore data for this Ligand-Target Pair
Affinity DataIC50: 0.770nMAssay Description:In vitro ability to inhibit the binding of [3H]spiperone to dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 0.810nMAssay Description:Displacement of [3H]methyl-spiperone from human recombinant D2S receptor in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Binding affinity against Dopamine receptor D2 from rat brain corpus striatum membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Displacement of [3H]raclopride from rat dopamine D2 receptorMore data for this Ligand-Target Pair