Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ic50 data for polymerid = 50004632
TargetC-C chemokine receptor type 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50382932(CHEMBL2029422)
Affinity DataIC50:  2.80nMAssay Description:Antagonist activity at rat CCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50337619(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxytetrahydr...)
Affinity DataIC50:  2.90nMAssay Description:Binding affinity to rat CCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50382932(CHEMBL2029422)
Affinity DataIC50:  13nMAssay Description:Binding affinity to rat CCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50385450(CHEMBL2036782)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at rat CCR2 receptor expressed in human THP-1 cells assessed as inhibition of MCP1-induced Ca2+ flux by FLIPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50331728(CHEMBL1289316 | N-(2-((3S,4S)-1-(cis-4-(benzo[d][1...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of rat CCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50339636(1-(6-((2-(Dimethylamino)ethyl)(methyl)amino)-1,3-d...)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity at CCR2 in rat spleen cells assessed as inhibition of CCL2-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed