Compile Data Set for Download or QSAR
maximum 50k data
Found 9 of ic50 data for polymerid = 50006192
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM50397589(CHEMBL2171517)
Affinity DataIC50:  5nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM50397590(CHEMBL2171516)
Affinity DataIC50:  20nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM50397588(CHEMBL2171518)
Affinity DataIC50:  60nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM50397592(CHEMBL2171514)
Affinity DataIC50:  240nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM50397593(CHEMBL2171513)
Affinity DataIC50:  260nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM50397591(CHEMBL2171515)
Affinity DataIC50:  510nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM47658(1-(4-methylphenyl)-3-(2-pyridin-3-ylpyrimidin-4-yl...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM50397595(CHEMBL2171512)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division related protein kinase 2(Leishmania major)
Montclair State University

Curated by ChEMBL
LigandPNGBDBM78336((6E)-6-[4-(3-pyridinylmethylamino)-1H-quinazolin-2...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of Leishmania major CRK3 expressed in Escherichia coli BL21 (DE3) using 5FAM-GGGRSPGRRRRK-OH as substrate after 60 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed