Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ic50 data for polymerid = 50006448
TargetBromodomain-containing protein 4(Mus musculus)
Icahn School Of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50443230(CHEMBL3086885)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of BRD4 in LPS-stimulated mouse RAW264.7 cells assessed as inhibition of NF-kappaB-mediated nitric oxide production preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Mus musculus)
Icahn School Of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50443230(CHEMBL3086885)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of BRD4 in LPS-stimulated mouse RAW264.7 cells assessed as inhibition of NF-kappaB-mediated IL-6 expression preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Mus musculus)
Icahn School Of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50443232(CHEMBL3086883)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of BRD4 in LPS-stimulated mouse RAW264.7 cells assessed as inhibition of NF-kappaB-mediated nitric oxide production preincubated for 30 mi...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Mus musculus)
Icahn School Of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50443232(CHEMBL3086883)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of BRD4 in LPS-stimulated mouse RAW264.7 cells assessed as inhibition of NF-kappaB-mediated IL-6 expression preincubated for 30 mins follo...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Mus musculus)
Icahn School Of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50443233(CHEMBL3087052)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of BRD4 in LPS-stimulated mouse RAW264.7 cells assessed as inhibition of NF-kappaB-mediated IL-6 expression preincubated for 30 mins follo...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Mus musculus)
Icahn School Of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50443231(CHEMBL3086884)
Affinity DataIC50:  2.32E+4nMAssay Description:Inhibition of BRD4 in LPS-stimulated mouse RAW264.7 cells assessed as inhibition of NF-kappaB-mediated IL-6 expression preincubated for 30 mins follo...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Mus musculus)
Icahn School Of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50443231(CHEMBL3086884)
Affinity DataIC50:  3.81E+4nMAssay Description:Inhibition of BRD4 in LPS-stimulated mouse RAW264.7 cells assessed as inhibition of NF-kappaB-mediated nitric oxide production preincubated for 30 mi...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Mus musculus)
Icahn School Of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50443233(CHEMBL3087052)
Affinity DataIC50:  4.63E+4nMAssay Description:Inhibition of BRD4 in LPS-stimulated mouse RAW264.7 cells assessed as inhibition of NF-kappaB-mediated nitric oxide production preincubated for 30 mi...More data for this Ligand-Target Pair