Affinity DataKd: 1.50E+3nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
Affinity DataKd: 7.10E+3nMAssay Description:Inhibition of human CYP3A4 assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 400nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
Affinity DataKd: 7.30E+3nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
Affinity DataKd: 2.30E+3nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
Affinity DataKd: 40nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
Affinity DataKd: 160nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
Affinity DataKd: 61nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 4 nM concentrationMore data for this Ligand-Target Pair
Affinity DataKd: 5.60nMAssay Description:Compound was evaluated for its effect towards [3H]-DPDPE binding to Opioid receptor delta 1 at 4 nM concentration expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 5.90nMAssay Description:Compound was evaluated for its effect towards [3H]-DPDPE binding to Opioid receptor delta 1 at 4 nM concentration expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 4 nM concentrationMore data for this Ligand-Target Pair
Affinity DataKd: 3.00E+4nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKd: 2.10nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKd: 4.00E+3nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 588nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 500nMAssay Description:Binding affinity to C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as spectral dissociatio...More data for this Ligand-Target Pair
Affinity DataKd: 900nMAssay Description:Binding affinity to C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as spectral dissociatio...More data for this Ligand-Target Pair
Affinity DataKd: 1.00E+4nMAssay Description:Binding affinity to C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as spectral dissociatio...More data for this Ligand-Target Pair
Affinity DataKd: 1.00E+4nMAssay Description:Binding affinity to C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as spectral dissociatio...More data for this Ligand-Target Pair
Affinity DataKd: 1.05E+5nMAssay Description:Binding affinity to C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as spectral dissociatio...More data for this Ligand-Target Pair
Affinity DataKd: 2.50E+6nMAssay Description:Binding affinity to C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as spectral dissociatio...More data for this Ligand-Target Pair
Affinity DataKd: 4.50E+6nMAssay Description:Binding affinity to C-terminal four-histidine tagged human CYP3A4delta3 to 24 residues expressed in Escherichia coli assessed as spectral dissociatio...More data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKd: 2.70E+3nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Affinity against the Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKd: 260nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 625nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 770nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 910nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 4.00E+3nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 715nMAssay Description:Binding affinity at Opioid receptor delta 1 in rat brain membrane was determined by using curve -fitting LIGAND([3H]DHM, [3H]DADL, [3H]DSLET, [3H]EKC...More data for this Ligand-Target Pair
Affinity DataKd: 40nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 0.25 nM concentrationMore data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Compound was evaluated for its effect towards [3H]-DPDPE binding to Opioid receptor delta 1 at 0.25 nM concentration expressed as dissociation consta...More data for this Ligand-Target Pair
Affinity DataKd: 4.30nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 4 nM concentrationMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Compound was evaluated for its effect towards [3H]-DPDPE binding to Opioid receptor delta 1 at 4 nM concentration expressed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 2.30nMAssay Description:Compound was evaluated for its effect towards [3H]-DSLET binding to Opioid receptor delta 2 at 4 nM concentrationMore data for this Ligand-Target Pair
Affinity DataKd: 3.00E+4nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 2.70E+3nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 4.00E+3nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 588nMAssay Description:Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGANDMore data for this Ligand-Target Pair
Affinity DataKd: 900nMAssay Description:Binding affinity to His-tagged CYP3A4 (unknown origin) expressed in Escherichia coli DH5alpha assessed as type 2 spectral shift by measuring dissocia...More data for this Ligand-Target Pair
Affinity DataKd: 1.60E+3nMAssay Description:Inhibition of human CYP3A4 assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 5.50E+3nMAssay Description:Inhibition of human CYP3A4 assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Inhibition of human CYP3A4 assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 370nMAssay Description:Inhibition of human CYP3A4 assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 1.31E+4nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair